XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 0.0 | 10 | uM |
| XMD8-92 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | -15.2 | 10 | uM |
| XMD8-92 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | -0.5 | 10 | uM |
| XMD8-92 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | -5.5 | 10 | uM |
| XMD8-92 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -15.9 | 10 | uM |
| XMD8-92 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 0.0 | 10 | uM |
| XMD8-92 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 9.1 | 10 | uM |
| XMD8-92 | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | 4.0 | 10 | uM |
| XMD8-92 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -5.5 | 10 | uM |
| XMD8-92 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | 5.6 | 10 | uM |
| XMD8-92 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -11.9 | 10 | uM |
| XMD8-92 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 5.0 | 10 | uM |
| XMD8-92 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -13.0 | 10 | uM |
| XMD8-92 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | 6.1 | 10 | uM |
| XMD8-92 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -2.3 | 10 | uM |
| XMD8-92 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 4.6 | 10 | uM |
| XMD8-92 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -7.3 | 10 | uM |
| XMD8-92 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -13.2 | 10 | uM |
| XMD8-92 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | 17.9 | 10 | uM |
| XMD8-92 | HeLa | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -24.6 | 10 | uM |
| XMD8-92 | PC-3 | CDK14 | LVALkVIR | Lys1 | -6.6 | 10 | uM |
| XMD8-92 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | -3.1 | 10 | uM |
| XMD8-92 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 6.0 | 10 | uM |
| XMD8-92 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 4.8 | 10 | uM |
| XMD8-92 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | 14.2 | 10 | uM |