XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | -2.2 | 10 | uM |
| XMD8-92 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | -1.3 | 10 | uM |
| XMD8-92 | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | 2.6 | 10 | uM |
| XMD8-92 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -11.5 | 10 | uM |
| XMD8-92 | HeLa | LYN | VAVkTLKPGTMSVQAFLEEANLMK | Lys1 | -6.0 | 10 | uM |
| XMD8-92 | PC-3 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -3.4 | 10 | uM |
| XMD8-92 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | -9.7 | 10 | uM |
| XMD8-92 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | 15.1 | 10 | uM |
| XMD8-92 | PC-3 | MARK2 | EVAVkIIDKTQLNSSSLQK | Lys1 | -4.9 | 10 | uM |
| XMD8-92 | PC-3 | MARK3,MARK4 | EVAIkIIDK | Lys1 | -17.9 | 10 | uM |
| XMD8-92 | HeLa | MASTL | LYAVkVVK | Lys1 | 8.9 | 10 | uM |
| XMD8-92 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | -10.5 | 10 | uM |
| XMD8-92 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 7.3 | 10 | uM |
| XMD8-92 | HeLa | p38a | DLkPSNLAVNEDCELK | Lys2 | -35.4 | 10 | uM |
| XMD8-92 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | -3.9 | 10 | uM |
| XMD8-92 | HeLa | MK14 | QELNkTIWEVPER | Other | 4.1 | 10 | uM |
| XMD8-92 | PC-3 | MK14 | QELNkTIWEVPER | Other | 13.3 | 10 | uM |
| XMD8-92 | HeLa | PAN3 | VMDPTkILITGK | -4.5 | 10 | uM | |
| XMD8-92 | HeLa | PEK | DLkPSNIFFTMDDVVK | Lys2 | -1.4 | 10 | uM |
| XMD8-92 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 5.1 | 10 | uM |
| XMD8-92 | HeLa | PIK3CG | KkPLWLEFK | ATP | -15.8 | 10 | uM |
| XMD8-92 | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | 17.4 | 10 | uM |
| XMD8-92 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 9.0 | 10 | uM |
| XMD8-92 | PC-3 | ROCK1 | kLQLELNQER | Other | -4.3 | 10 | uM |
| XMD8-92 | PC-3 | RON | IQCAIkSLSR | Lys1 | -5.6 | 10 | uM |