JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JWE-035 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 91.1 | 10 | uM |
| JWE-035 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 30.9 | 10 | uM |
| JWE-035 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -18.2 | 10 | uM |
| JWE-035 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 63.0 | 10 | uM |
| JWE-035 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 57.2 | 10 | uM |
| JWE-035 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 55.4 | 10 | uM |
| JWE-035 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 75.7 | 10 | uM |
| JWE-035 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | 7.3 | 10 | uM |
| JWE-035 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 6.2 | 10 | uM |
| JWE-035 | PC-3 | ATR | FYIMMCkPK | ATP | 3.6 | 10 | uM |
| JWE-035 | HeLa | ATR | FYIMMCkPK | ATP | 8.1 | 10 | uM |
| JWE-035 | HeLa | AurB | SHFIVALkVLFK | Lys1 | 80.4 | 10 | uM |
| JWE-035 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 4.4 | 10 | uM |
| JWE-035 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 4.5 | 10 | uM |
| JWE-035 | HeLa | BTK | GQYDVAIkMIK | Lys1 | 2.0 | 10 | uM |
| JWE-035 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 0.8 | 10 | uM |
| JWE-035 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | 2.2 | 10 | uM |
| JWE-035 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | -3.2 | 10 | uM |
| JWE-035 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 21.0 | 10 | uM |
| JWE-035 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.9 | 10 | uM |
| JWE-035 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 16.0 | 10 | uM |
| JWE-035 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 12.9 | 10 | uM |
| JWE-035 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 0.7 | 10 | uM |
| JWE-035 | PC-3 | CDK14 | LVALkVIR | Lys1 | 14.6 | 10 | uM |
| JWE-035 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | 2.7 | 10 | uM |