JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JWE-035 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | 16.8 | 10 | uM |
| JWE-035 | HeLa | SYK | ISDFGLSkALR | Activation Loop | -0.1 | 10 | uM |
| JWE-035 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | -43.4 | 10 | uM |
| JWE-035 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | 5.8 | 10 | uM |
| JWE-035 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | 12.8 | 10 | uM |
| JWE-035 | HeLa | RSK1 domain1 | LTDFGLSkEAIDHEK | Activation Loop | -9.4 | 10 | uM |
| JWE-035 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -6.1 | 10 | uM |
| JWE-035 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 16.2 | 10 | uM |
| JWE-035 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | -6.9 | 10 | uM |
| JWE-035 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 30.0 | 10 | uM |
| JWE-035 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 12.3 | 10 | uM |
| JWE-035 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 22.4 | 10 | uM |
| JWE-035 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | 28.3 | 10 | uM |
| JWE-035 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | 3.5 | 10 | uM |
| JWE-035 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | 91.1 | 10 | uM |
| JWE-035 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 3.2 | 10 | uM |
| JWE-035 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | 75.6 | 10 | uM |
| JWE-035 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -0.3 | 10 | uM |
| JWE-035 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -10.2 | 10 | uM |
| JWE-035 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 41.6 | 10 | uM |
| JWE-035 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 1.4 | 10 | uM |
| JWE-035 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -19.5 | 10 | uM |
| JWE-035 | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | 23.9 | 10 | uM |
| JWE-035 | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | 12.1 | 10 | uM |
| JWE-035 | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 27.9 | 10 | uM |