JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
JWE-035 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -13.3 | 10 | uM |
JWE-035 | PC-3 | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 26.4 | 10 | uM |
JWE-035 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 16.9 | 10 | uM |
JWE-035 | HeLa | IRAK3 | SHLEHQSCTINMTSSSSkHLWYMPEEYIR | Protein Kinase Domain | 33.0 | 10 | uM |
JWE-035 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.9 | 10 | uM |
JWE-035 | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 8.5 | 10 | uM |
JWE-035 | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | -48.5 | 10 | uM |
JWE-035 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | -401.7 | 10 | uM |
JWE-035 | HeLa | MK14 | QELNkTIWEVPER | Other | 7.9 | 10 | uM |
JWE-035 | PC-3 | ROCK1 | kLQLELNQER | Other | 18.7 | 10 | uM |
JWE-035 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 7.3 | 10 | uM |
JWE-035 | PC-3 | MK14 | QELNkTIWEVPER | Other | -5.9 | 10 | uM |
JWE-035 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 93.2 | 10 | uM |
JWE-035 | PC-3 | MK11 | QELNkTVWEVPQR | Other | -14.7 | 10 | uM |
JWE-035 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -1.7 | 10 | uM |
JWE-035 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 7.2 | 10 | uM |
JWE-035 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | 10.5 | 10 | uM |
JWE-035 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 7.1 | 10 | uM |
JWE-035 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -0.4 | 10 | uM |
JWE-035 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -5.7 | 10 | uM |
JWE-035 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 29.0 | 10 | uM |
JWE-035 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 4.5 | 10 | uM |
JWE-035 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | 4.2 | 10 | uM |
JWE-035 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | 4.2 | 10 | uM |
JWE-035 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | 54.2 | 10 | uM |