PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

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Small Molecule Cell Line Protein Sequence Labeling Site IC50 Conc unit
PLX-4720 A-375 PKN2
DLkLDNLLLDTEGFVK
LYS2
>10
uM
PLX-4720 A-375 PKR
DLkPSNIFLVDTK
LYS2
>10
uM
PLX-4720 A-375 PLK1
CFEISDADTKEVFAGkIVPK
LYS1
>10
uM
PLX-4720 A-375 PRKACB
DLkPENLLIDHQGYIQ
LYS2
>10
uM
PLX-4720 A-375 PRPK
FLSGLELVkQGAEAR
ATP Loop
>10
uM
PLX-4720 A-375 RAF1
DMkSNNIFLHEGLTVK
LYS2
0.35
uM
PLX-4720 A-375 ROCK1,ROCK2
DVkPDNMLLDK
LYS2
>10
uM
PLX-4720 A-375 RSK1,RSK2,RSK3_domain1
DLkPENILLDEEGHIK
LYS2
>10
uM
PLX-4720 A-375 RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
LYS2
>10
uM
PLX-4720 A-375 RSK1_domain1
LTDFGLSkEAIDHEKK
Activation Loop
>10
uM
PLX-4720 A-375 RSK1_domain1
KVTRPDSGHLYAMkVLK
LYS1
>10
uM
PLX-4720 A-375 RSK1_domain2
DLkPSNILYVDESGNPECLR
LYS2
>10
uM
PLX-4720 A-375 RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
>10
uM
PLX-4720 A-375 RSK2_domain2
DLkPSNILYVDESGNPESIR
LYS2
>10
uM
PLX-4720 A-375 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
>10
uM
PLX-4720 A-375 RSK2_domain2
TVEYLHAQGVVHRDLkPSNILYVDESGNPESIR
LYS2
>10
uM
PLX-4720 A-375 RSK3_domain1
DLkPENILLDEEGHIKITDFGLSK
LYS2
>10
uM
PLX-4720 A-375 RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
>10
uM
PLX-4720 A-375 SGK3
FYAVkVLQK
LYS1
11.0
uM
PLX-4720 A-375 SLK
AQNKETSVLAAAkVIDTK
LYS1
>10
uM
PLX-4720 A-375 SLK
IIHRDLkAGNILFTLDGDIK
LYS2
>10
uM
PLX-4720 A-375 SLK
DLkAGNILFTLDGDIK
LYS2
>10
uM
PLX-4720 A-375 SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
>10
uM
PLX-4720 A-375 SRC
VAIkTLKPGTMSPEAFLQEAQVMKK
LYS1
4.7
uM
PLX-4720 A-375 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
LYS1
3.5
uM