PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

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Small Molecule Cell Line Protein Sequence Labeling Site IC50 Conc unit
PLX-4720 A-375 RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
>10
uM
PLX-4720 A-375 PI4KB
VPHTQAVVLNSkDK
ATP
>10
uM
PLX-4720 A-375 PI4KB
VPHTQAVVLNSKDkAPYLIYVEVLECENFDTTSVPAR
ATP
>10
uM
PLX-4720 A-375 GCN2_domain2
VQNKLDGCCYAVkR
LYS1
3.9
uM
PLX-4720 A-375 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
6.4
uM
PLX-4720 A-375 CSK
VSDFGLTkEASSTQDTGKLPVKWTAPEALR
Activation Loop
6.1
uM
PLX-4720 A-375 MLTK
WISQDKEVAVKk
LYS1
0.011
uM
PLX-4720 A-375 ILK
WQGNDIVVkVLK
LYS1
>10
uM
PLX-4720 A-375 JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
LYS1
>10
uM
PLX-4720 A-375 MK03
YIHSANVLHRDLkPSNLLINTTCDLK
LYS2
>10
uM
PLX-4720 A-375 WEE1
YIHSMSLVHMDIkPSNIFISR
LYS2
>10
uM
PLX-4720 A-375 eEF2K
YIkYNSNSGFVR
ATP
>10
uM
PLX-4720 A-375 eEF2K
YIkYNSNSGFVRDDNIR
ATP
>10
uM
PLX-4720 A-375 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
LYS2
>10
uM
PLX-4720 A-375 ABL,ARG
YSLTVAVkTLKEDTMEVEEFLK
LYS1
0.33
uM
PLX-4720 A-375 STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
>10
uM
PLX-4720 A-375 TLK2
YVAVkIHQLNK
LYS1
>10
uM