PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

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Small Molecule Cell Line Protein Sequence Labeling Site IC50 Conc unit
PLX-4720 A-375 RSK2_domain2
TVEYLHAQGVVHRDLkPSNILYVDESGNPESIR
LYS2
>10
uM
PLX-4720 A-375 RSK3_domain1
DLkPENILLDEEGHIKITDFGLSK
LYS2
>10
uM
PLX-4720 A-375 SLK
IIHRDLkAGNILFTLDGDIK
LYS2
>10
uM
PLX-4720 A-375 SLK
DLkAGNILFTLDGDIK
LYS2
>10
uM
PLX-4720 A-375 TAO1,TAOK3
DIkAGNILLTEPGQVK
LYS2
>10
uM
PLX-4720 A-375 TAOK2
DVkAGNILLSEPGLVK
LYS2
>10
uM
PLX-4720 A-375 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
LYS2
>10
uM
PLX-4720 A-375 ULK3
NISHLDLkPQNILLSSLEKPHLK
LYS2
>10
uM
PLX-4720 A-375 VRK2
MLDVLEYIHENEYVHGDIkAANLLLGYK
LYS2
>10
uM
PLX-4720 A-375 WEE1
YIHSMSLVHMDIkPSNIFISR
LYS2
>10
uM
PLX-4720 A-375 Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
LYS2
>10
uM
PLX-4720 A-375 WNK4
DLkCDNVFITGPTGSVK
LYS2
>10
uM
PLX-4720 A-375 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
LYS2
2.0
uM
PLX-4720 A-375 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
>10
uM
PLX-4720 A-375 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
>10
uM
PLX-4720 A-375 JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Protein Kinase Domain
>10
uM
PLX-4720 A-375 RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
>10
uM