PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | IC50 | Conc unit |
|---|---|---|---|---|---|---|
| PLX-4720 | A-375 | GCN2_domain2 | VQNKLDGCCYAVkR | LYS1 | 3.9 | uM |
| PLX-4720 | A-375 | NEK7 | AACLLDGVPVALkK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | CDK5 | NRETHEIVALkR | LYS1 | >10 | uM |
| PLX-4720 | A-375 | NDR2 | KDTGHIYAMkILR | LYS1 | >10 | uM |
| PLX-4720 | A-375 | GCK | DTVTSELAAVkIVK | LYS1 | 4.0 | uM |
| PLX-4720 | A-375 | FER | TSVAVkTCKEDLPQELK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | FER | DKTSVAVkTCKEDLPQELK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | NDR2 | DTGHIYAMkILR | LYS1 | >10 | uM |
| PLX-4720 | A-375 | NDR1 | DTGHVYAMkILR | LYS1 | >10 | uM |
| PLX-4720 | A-375 | ACK | TVSVAVKCLkPDVLSQPEAMDDFIR | LYS1 | 0.22 | uM |
| PLX-4720 | A-375 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | NEK9 | TEDDSLVVWkEVDLTR | LYS1 | >10 | uM |
| PLX-4720 | A-375 | CDK2 | NKLTGEVVALkK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | MST1 | AIHKETGQIVAIkQVPVESDLQEIIK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | ABL,ARG | YSLTVAVkTLKEDTMEVEEFLK | LYS1 | 0.33 | uM |
| PLX-4720 | A-375 | MST1 | ETGQIVAIkQVPVESDLQEIIK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | MST2 | ESGQVVAIkQVPVESDLQEIIK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | NDR1 | KDTGHVYAMkILR | LYS1 | >10 | uM |
| PLX-4720 | A-375 | EGFR | IPVAIkELR | LYS1 | >10 | uM |
| PLX-4720 | A-375 | CaMKK2 | LAYNENDNTYYAMkVLSK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | CASK | ETGQQFAVkIVDVAK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | MLKL | APVAIkVFK | LYS1 | 4.9 | uM |
| PLX-4720 | A-375 | CaMK2g | KTSTQEYAAkIINTKK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | MAP3K3 | ELASkQVQFDPDSPETSKEVSALECEIQLLK | LYS1 | >10 | uM |
| PLX-4720 | A-375 | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | LYS1 | >10 | uM |