PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

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Small Molecule Cell Line Protein Sequence Labeling Site IC50 Conc unit
PLX-4720 A-375 CDK5
NRETHEIVALkR
LYS1
>10
uM
PLX-4720 A-375 CDK2
NKLTGEVVALkK
LYS1
>10
uM
PLX-4720 A-375 LOK
NKETGALAAAkVIETK
LYS1
>10
uM
PLX-4720 A-375 PKD3
NIVHCDLkPENVLLASAEPFPQVK
LYS2
>10
uM
PLX-4720 A-375 PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
LYS2
>10
uM
PLX-4720 A-375 ULK3
NISHLDLkPQNILLSSLEKPHLK
LYS2
>10
uM
PLX-4720 A-375 AXL
NCMLNENMSVCVADFGLSkK
Activation Loop
>10
uM
PLX-4720 A-375 MAP2K4
MVHKPSGQIMAVkR
LYS1
5.6
uM
PLX-4720 A-375 VRK2
MLDVLEYIHENEYVHGDIkAANLLLGYK
LYS2
>10
uM
PLX-4720 A-375 MAP2K6
MCDFGISGYLVDSVAkTIDAGCKPYMAPER
Activation Loop
>10
uM
PLX-4720 A-375 CDK14
LVALkVIR
LYS1
>10
uM
PLX-4720 A-375 CaMK1a
LVAIkCIAK
LYS1
13.0
uM
PLX-4720 A-375 CDK16
LTDNLVALkEIR
LYS1
>10
uM
PLX-4720 A-375 RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
>10
uM
PLX-4720 A-375 RSK1_domain1
LTDFGLSkEAIDHEKK
Activation Loop
>10
uM
PLX-4720 A-375 KS6B2
LTDFGLCkESIHEGAVTHTFCGTIEYMAPEILVR
Activation Loop
>10
uM
PLX-4720 A-375 KS6B1
LTDFGLCkESIHDGTVTHTFCGTIEYMAPEILMR
Activation Loop
>10
uM
PLX-4720 A-375 NDR1,NDR2
LSDFGLCTGLkK
Activation Loop
>10
uM
PLX-4720 A-375 ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
0.83
uM
PLX-4720 A-375 NEK9
LGDYGLAkK
Activation Loop
>10
uM
PLX-4720 A-375 CaMKK2
LAYNENDNTYYAMkVLSK
LYS1
>10
uM
PLX-4720 A-375 MST3,MST4,YSK1
LADFGVAGQLTDTQIkR
Activation Loop
>10
uM
PLX-4720 A-375 RSK1_domain1
KVTRPDSGHLYAMkVLK
LYS1
>10
uM
PLX-4720 A-375 CaMK2g
KTSTQEYAAkIINTKK
LYS1
>10
uM
PLX-4720 A-375 MAP2K1,MAP2K2
kLIHLEIKPAIR
LYS1
>10
uM