PLX-4720 KiNativ -- dose response experiment - Dataset (ID:20090)

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Small Molecule Cell Line Protein Sequence Labeling Site IC50 Conc unit
PLX-4720 A-375 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
>10
uM
PLX-4720 A-375 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
6.4
uM
PLX-4720 A-375 AXL
NCMLNENMSVCVADFGLSkK
Activation Loop
>10
uM
PLX-4720 A-375 NDR1,NDR2
LSDFGLCTGLkK
Activation Loop
>10
uM
PLX-4720 A-375 MAP2K6
MCDFGISGYLVDSVAkTIDAGCKPYMAPER
Activation Loop
>10
uM
PLX-4720 A-375 CSK
VSDFGLTkEASSTQDTGKLPVKWTAPEALR
Activation Loop
6.1
uM
PLX-4720 A-375 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
>10
uM
PLX-4720 A-375 KS6B2
LTDFGLCkESIHEGAVTHTFCGTIEYMAPEILVR
Activation Loop
>10
uM
PLX-4720 A-375 RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
>10
uM
PLX-4720 A-375 JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
>10
uM
PLX-4720 A-375 KS6B1
LTDFGLCkESIHDGTVTHTFCGTIEYMAPEILMR
Activation Loop
>10
uM
PLX-4720 A-375 ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
0.83
uM
PLX-4720 A-375 NEK9
LGDYGLAkK
Activation Loop
>10
uM
PLX-4720 A-375 RSK1_domain1
LTDFGLSkEAIDHEKK
Activation Loop
>10
uM
PLX-4720 A-375 NEK7
FFSSkTTAAHSLVGTPYYMSPER
Activation Loop
>10
uM
PLX-4720 A-375 STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
>10
uM
PLX-4720 A-375 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
6.2
uM