Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
MDA-MB-436 | Cediranib | 10.0 | VEGFR/cKIT | RTK | -0.3824 | 0.39722 |
CAMA-1 | Volasertib | 0.1 | PLK | Cell cycle | -0.3812 | 0.53477 |
CAMA-1 | Etoposide | 3.1623 | Topo II | Chemotherapy | -0.3802 | 0.45373 |
SUM159PT | Ceritinib | 10.0 | ALK | RTK | -0.3800 | 0.80163 |
CAMA-1 | Dinaciclib | 0.1 | pan CDK | Cell cycle | -0.3799 | 0.45483 |
MDA-MB-468 | Volasertib | 0.01 | PLK | Cell cycle | -0.3797 | 0.64007 |
CAL-85-1 | Luminespib | 0.1 | HSP90 | Misc | -0.3793 | 0.56133 |
HCC1954 | Buparlisib | 3.1623 | pan PI3K | PI3K/mTOR | -0.3790 | 0.64694 |
CAL-85-1 | Doxorubicin | 1.0 | Chemo | Chemotherapy | -0.3783 | 0.43963 |
SUM149PT | Luminespib | 0.1 | HSP90 | Misc | -0.3767 | 0.68080 |
CAL-85-1 | Luminespib | 0.31623 | HSP90 | Misc | -0.3765 | 0.56828 |
HCC1428 | Topotecan | 10.0 | Topo I | Chemotherapy | -0.3764 | 0.49642 |
HCC1806 | AZD7762 | 3.1623 | CHK1/2 | Cell cycle | -0.3761 | 0.66396 |
Hs 578T | Taxol | 1.0 | Chemo | Chemotherapy | -0.3752 | 0.74970 |
BT-20 | Taselisib | 10.0 | PI3Ka, g, d | PI3K/mTOR | -0.3749 | 0.60583 |
HCC1954 | Luminespib | 1.0 | HSP90 | Misc | -0.3745 | 0.65805 |
HCC38 | Dinaciclib | 0.031623 | pan CDK | Cell cycle | -0.3744 | 0.44124 |
SUM149PT | Luminespib | 0.31623 | HSP90 | Misc | -0.3744 | 0.67001 |
MDA-MB-361 | AZD7762 | 0.1 | CHK1/2 | Cell cycle | -0.3743 | 0.24817 |
MDA-MB-453 | Pictilisib | 10.0 | pan PI3K | PI3K/mTOR | -0.3736 | 0.38023 |
MDA-MB-361 | AZD7762 | 3.1623 | CHK1/2 | Cell cycle | -0.3733 | 0.23979 |
SK-BR-3 | Buparlisib | 10.0 | pan PI3K | PI3K/mTOR | -0.3731 | 0.45147 |
PDXHCI002 | Tivantinib | 1.0 | MET | RTK | -0.3731 | 0.60360 |
CAL-85-1 | Luminespib | 0.031623 | HSP90 | Misc | -0.3724 | 0.57889 |
HCC1419 | Torin2 | 1.0 | mTOR/ATM/ATR | PI3K/mTOR | -0.3722 | 0.38672 |