Growth rate-corrected (GR) dose-response metrics across a panel of 71 breast cancer cell lines treated with a library of small molecule and antibody perturbagens. Dataset 1 of 4: Relative cell counts and normalized growth rate inhibition values across technical replicates. - Dataset (ID:20268)
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Cell | Clinical Subtype | Transcriptional Subtype | Small Molecule | Antibody | Perturbagen Target | Perturbagen Class | Perturbagen Concentration | Perturbagen Conc Unit | Biological Replicate ID | Relative Cell Count | Normalized Growth Rate Inhibition Value | Nominal Division Rate |
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184A1 | NM | Basal | AS-252424 | PI3K | PI3K | 6.67 | uM | 12509.165 | 0.5506 | 0.3443 | 1.5022 | |
184A1 | NM | Basal | Baicalein | Lipoxygenase | Metabolism | 0.000427 | uM | 5895.073 | 1.0365 | 1.0503 | 1.4431 | |
184A1 | NM | Basal | Baicalein | Lipoxygenase | Metabolism | 0.00213 | uM | 5895.073 | 1.0337 | 1.0465 | 1.4431 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 0.267 | uM | 9047.132 | 0.9995 | 0.9985 | 0.6985 | ||
184A1 | NM | Basal | 5-FU | TYMS | TYMS | 3840 | uM | 9047.017 | 0.1150 | -0.8459 | 0.8440 | |
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 0.000171 | uM | 12509.165 | 0.9871 | 0.9828 | 1.5022 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.00128 | uM | 9047.037 | 1.0758 | 1.2981 | 0.5262 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 0.000427 | uM | 9047.132 | 1.0270 | 1.0778 | 0.6985 | ||
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 0.0213 | uM | 12509.165 | 0.5575 | 0.3556 | 1.5022 | |
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 0.533 | uM | 12509.165 | 0.3318 | -0.0404 | 1.5022 | |
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 0.107 | uM | 12509.165 | 0.3373 | -0.0298 | 1.5022 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 0.00213 | uM | 9047.132 | 0.9693 | 0.9128 | 0.6985 | ||
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 66.7 | uM | 12509.165 | 0.0097 | -0.9088 | 1.5022 | |
184A1 | NM | Basal | Baicalein | Lipoxygenase | Metabolism | 33.3 | uM | 5895.073 | 0.8615 | 0.8038 | 1.4431 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.000256 | uM | 9047.037 | 0.9096 | 0.6705 | 0.5262 | |
184A1 | NM | Basal | AG1024 | IGF1R | RTK | 0.000427 | uM | 5894.066 | 1.0325 | 1.0430 | 1.5027 | |
184A1 | NM | Basal | Bortezomib | Proteasome | Proteasome | 0.000427 | uM | 5894.074 | 1.0584 | 1.0796 | 1.4541 | |
184A1 | NM | Basal | AG1024 | IGF1R | RTK | 0.0000853 | uM | 5894.066 | 1.0769 | 1.1011 | 1.5027 | |
184A1 | NM | Basal | Bortezomib | Proteasome | Proteasome | 0.00213 | uM | 5894.074 | 1.0465 | 1.0635 | 1.4541 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 1.33 | uM | 9047.132 | 0.9661 | 0.9036 | 0.6985 | ||
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.8 | uM | 9047.037 | 0.4311 | -0.5959 | 0.5262 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 4 | uM | 9047.037 | 0.4226 | -0.6108 | 0.5262 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.032 | uM | 9047.037 | 0.4452 | -0.5704 | 0.5262 | |
184A1 | NM | Basal | Bortezomib | Proteasome | Proteasome | 0.000427 | uM | 5895.074 | 1.0527 | 1.0937 | 1.1218 | |
184A1 | NM | Basal | Bortezomib | Proteasome | Proteasome | 167 | uM | 5894.074 | 0.0861 | -0.6297 | 1.4541 |