Growth rate-corrected (GR) dose-response metrics across a panel of 71 breast cancer cell lines treated with a library of small molecule and antibody perturbagens. Dataset 1 of 4: Relative cell counts and normalized growth rate inhibition values across technical replicates. - Dataset (ID:20268)

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Cell Clinical Subtype Transcriptional Subtype Small Molecule Antibody Perturbagen Target Perturbagen Class Perturbagen Concentration Perturbagen Conc Unit Biological Replicate ID Relative Cell Count Normalized Growth Rate Inhibition Value Nominal Division Rate
184A1
NM
Basal
AS-252424
PI3K
PI3K
6.67
uM
12509.165
0.5506 0.3443 1.5022
184A1
NM
Basal
Baicalein
Lipoxygenase
Metabolism
0.000427
uM
5895.073
1.0365 1.0503 1.4431
184A1
NM
Basal
Baicalein
Lipoxygenase
Metabolism
0.00213
uM
5895.073
1.0337 1.0465 1.4431
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
0.267
uM
9047.132
0.9995 0.9985 0.6985
184A1
NM
Basal
5-FU
TYMS
TYMS
3840
uM
9047.017
0.1150 -0.8459 0.8440
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
0.000171
uM
12509.165
0.9871 0.9828 1.5022
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.00128
uM
9047.037
1.0758 1.2981 0.5262
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
0.000427
uM
9047.132
1.0270 1.0778 0.6985
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
0.0213
uM
12509.165
0.5575 0.3556 1.5022
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
0.533
uM
12509.165
0.3318 -0.0404 1.5022
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
0.107
uM
12509.165
0.3373 -0.0298 1.5022
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
0.00213
uM
9047.132
0.9693 0.9128 0.6985
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
66.7
uM
12509.165
0.0097 -0.9088 1.5022
184A1
NM
Basal
Baicalein
Lipoxygenase
Metabolism
33.3
uM
5895.073
0.8615 0.8038 1.4431
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.000256
uM
9047.037
0.9096 0.6705 0.5262
184A1
NM
Basal
AG1024
IGF1R
RTK
0.000427
uM
5894.066
1.0325 1.0430 1.5027
184A1
NM
Basal
Bortezomib
Proteasome
Proteasome
0.000427
uM
5894.074
1.0584 1.0796 1.4541
184A1
NM
Basal
AG1024
IGF1R
RTK
0.0000853
uM
5894.066
1.0769 1.1011 1.5027
184A1
NM
Basal
Bortezomib
Proteasome
Proteasome
0.00213
uM
5894.074
1.0465 1.0635 1.4541
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
1.33
uM
9047.132
0.9661 0.9036 0.6985
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.8
uM
9047.037
0.4311 -0.5959 0.5262
184A1
NM
Basal
17-AAG
HSP90
HSP90
4
uM
9047.037
0.4226 -0.6108 0.5262
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.032
uM
9047.037
0.4452 -0.5704 0.5262
184A1
NM
Basal
Bortezomib
Proteasome
Proteasome
0.000427
uM
5895.074
1.0527 1.0937 1.1218
184A1
NM
Basal
Bortezomib
Proteasome
Proteasome
167
uM
5894.074
0.0861 -0.6297 1.4541