DCC-2036 KiNativ -- single dose experiment - Dataset (ID:20210)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| DCC-2036 | Ramos (RA 1) | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 18.5 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -19.6 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | ULK3 | EVVAIKCVAK | Lys1 | -25.3 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | MLTK | WISQDKEVAVKK | Lys1 | 80.7 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 72.4 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | 76.4 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | KCC2D | IPTGQEYAAKIINTKK | Lys1 | -4.2 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | KC1G1 | DVKPENFLIGR | Lys2 | 8.4 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 20.1 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | 75.4 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | MARK1,MARK2 | EVAVKIIDK | Lys1 | -16.2 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | KPCI | DLKLDNVLLDSEGHIK | Lys2 | -16.0 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | ZAP70 | ISDFGLSKALGADDSYYTAR | Activation Loop | 3.9 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | KCC4 | DLKPENLLYATPAPDAPLK | Lys2 | 33.9 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | MK01 | DLKPSNLLLNTTCDLK | Lys2 | -17.9 | 1 | uM |
| DCC-2036 | Ramos (RA 1) | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | 30.4 | 1 | uM |