DCC-2036 KiNativ -- single dose experiment - Dataset (ID:20210)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
DCC-2036 Ramos (RA 1) FRAP1
IQSIAPSLQVITSKQRPR
ATP
-15.1
 1
uM
DCC-2036 Ramos (RA 1) FYN,SRC,YES
QGAKFPIKWTAPEAALYGR
Activation Loop
39.2
 1
uM
DCC-2036 Ramos (RA 1) GCK
DIKGANLLLTLQGDVK
Lys2
26.1
 1
uM
DCC-2036 Ramos (RA 1) GSK3A
DIKPQNLLVDPDTAVLK
Lys2
5.4
 1
uM
DCC-2036 Ramos (RA 1) GSK3B
DIKPQNLLLDPDTAVLK
Lys2
32.9
 1
uM
DCC-2036 Ramos (RA 1) HPK1
DKVSGDLVALKMVK
Lys1
1.8
 1
uM
DCC-2036 Ramos (RA 1) IKKE
SGELVAVKVFNTTSYLRPR
Lys1
-0.9
 1
uM
DCC-2036 Ramos (RA 1) IKKE,TBK1
DIKPGNIMR
Lys2
7.2
 1
uM
DCC-2036 Ramos (RA 1) ILK
ISMADVKFSFQCPGR
Protein Kinase Domain
-26.6
 1
uM
DCC-2036 Ramos (RA 1) IRAK4
DIKSANILLDEAFTAK
Lys2
33.1
 1
uM
DCC-2036 Ramos (RA 1) JAK1
QLASALSYLEDKDLVHGNVCTKNLLLAR
Protein Kinase Domain
29.6
 1
uM
DCC-2036 Ramos (RA 1) JAK1_domain2
YDPEGDNTGEQVAVKSLKPESGGNHIADLKK
Lys1
19.3
 1
uM
DCC-2036 Ramos (RA 1) JNK1,JNK2,JNK3
DLKPSNIVVK
Lys2
10.7
 1
uM
DCC-2036 Ramos (RA 1) KHS1
NVHTGELAAVKIIK
Lys1
-13.0
 1
uM
DCC-2036 Ramos (RA 1) LKB1
DIKPGNLLLTTGGTLK
Lys2
-2.5
 1
uM
DCC-2036 Ramos (RA 1) LOK
DLKAGNVLMTLEGDIR
Lys2
63.0
 1
uM
DCC-2036 Ramos (RA 1) LYN
VAVKTLKPGTMSVQAFLEEANLMK
Lys1
90.7
 1
uM
DCC-2036 Ramos (RA 1) LYN
EGAKFPIKWTAPEAINFGCFTIK
Activation Loop
79.6
 1
uM
DCC-2036 Ramos (RA 1) MAP2K1
IMHRDVKPSNILVNSR
Lys2
-11.8
 1
uM
DCC-2036 Ramos (RA 1) MAP2K1,MAP2K2
DVKPSNILVNSR
Lys2
0.4
 1
uM
DCC-2036 Ramos (RA 1) MAP2K3
DVKPSNVLINK
Lys2
-10.2
 1
uM
DCC-2036 Ramos (RA 1) MAP2K4
DIKPSNILLDR
Lys2
-8.7
 1
uM
DCC-2036 Ramos (RA 1) MAP2K5
DVKPSNMLVNTR
Lys2
4.9
 1
uM
DCC-2036 Ramos (RA 1) MAP2K6
DVKPSNVLINALGQVK
Lys2
-2.1
 1
uM
DCC-2036 Ramos (RA 1) MP2K7
DVKPSNILLDER
Lys2
-0.7
 1
uM