Gefitinib KINOMEscan - Dataset (ID:20161)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Gefitinib | EGFR(L747-T751del,Sins) | 0.5 | nM |
Gefitinib | EGFR(E746-A750del) | 0.5 | nM |
Gefitinib | EGFR(L747-S752del, P753S) | 0.6 | nM |
Gefitinib | EGFR(L747-E749del, A750P) | 0.6 | nM |
Gefitinib | EGFR(L858R) | 0.9 | nM |
Gefitinib | EGFR | 1.0 | nM |
Gefitinib | EGFR(S752-I759del) | 1.0 | nM |
Gefitinib | EGFR(G719S) | 1.1 | nM |
Gefitinib | EGFR(L861Q) | 1.4 | nM |
Gefitinib | EGFR(G719C) | 2.0 | nM |
Gefitinib | GAK | 13.0 | nM |
Gefitinib | EGFR(T790M) | 40.0 | nM |
Gefitinib | IRAK1 | 69.0 | nM |
Gefitinib | EGFR(L858R,T790M) | 140.0 | nM |
Gefitinib | ABL1(Q252H)-phosphorylated | 230.0 | nM |
Gefitinib | YSK4 | 240.0 | nM |
Gefitinib | MKNK1 | 290.0 | nM |
Gefitinib | HIPK4 | 310.0 | nM |
Gefitinib | ABL1(Y253F)-phosphorylated | 360.0 | nM |
Gefitinib | ABL1(E255K)-phosphorylated | 400.0 | nM |
Gefitinib | ERBB4 | 410.0 | nM |
Gefitinib | CSNK1E | 430.0 | nM |
Gefitinib | ABL1(H396P)-phosphorylated | 460.0 | nM |
Gefitinib | LOK | 470.0 | nM |
Gefitinib | ABL1-phosphorylated | 480.0 | nM |