Gefitinib KINOMEscan - Dataset (ID:20161)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Gefitinib | AAK1 | nM | |
| Gefitinib | ABL1(E255K)-phosphorylated | 400.0 | nM |
| Gefitinib | ABL1(F317I)-nonphosphorylated | nM | |
| Gefitinib | ABL1(F317I)-phosphorylated | 4700.0 | nM |
| Gefitinib | ABL1(F317L)-nonphosphorylated | 2700.0 | nM |
| Gefitinib | ABL1(F317L)-phosphorylated | 780.0 | nM |
| Gefitinib | ABL1(H396P)-nonphosphorylated | 680.0 | nM |
| Gefitinib | ABL1(H396P)-phosphorylated | 460.0 | nM |
| Gefitinib | ABL1(M351T)-phosphorylated | 520.0 | nM |
| Gefitinib | ABL1(Q252H)-nonphosphorylated | 1100.0 | nM |
| Gefitinib | ABL1(Q252H)-phosphorylated | 230.0 | nM |
| Gefitinib | ABL1(T315I)-nonphosphorylated | nM | |
| Gefitinib | ABL1(T315I)-phosphorylated | nM | |
| Gefitinib | ABL1(Y253F)-phosphorylated | 360.0 | nM |
| Gefitinib | ABL1-nonphosphorylated | 2200.0 | nM |
| Gefitinib | ABL1-phosphorylated | 480.0 | nM |
| Gefitinib | ABL2 | 1600.0 | nM |
| Gefitinib | ACVR1 | nM | |
| Gefitinib | ACVR1B | nM | |
| Gefitinib | ACVR2A | nM | |
| Gefitinib | ACVR2B | nM | |
| Gefitinib | ACVRL1 | nM | |
| Gefitinib | ADCK3 | nM | |
| Gefitinib | ADCK4 | nM | |
| Gefitinib | AKT1 | nM |