Breast cell line dose response to target inhibition measured by high throughput microscopy - Dataset (ID:20136)
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Small Molecule | Cell Line | Drug Concentration | Conc Units | Timepoint | Timepoint Units | Measured pERK (Alexa 488) | Measured p-Rb (Alexa 568) | Alexa Fluor 647 | Measured p-Akt/p-4EBP1/p-S6 (Alexa 647) | Image |
---|---|---|---|---|---|---|---|---|---|---|
Gefitinib | T47D | 0 (control) | 24 | hr | 177.88 | 116.19 | p-Akt | 85.23 | ||
Dactolisib | T47D | 0 (control) | 24 | hr | 165.27 | 86.01 | p-Akt | 60.10 | ||
GSK1059615 | MCF 10A | 0 (control) | 24 | hr | 372.12 | 121.72 | p-Akt | 53.36 | ||
Dactolisib | MCF 10A | 0 (control) | 24 | hr | 351.94 | 125.18 | p-Akt | 50.36 | ||
GSK1059615 | T47D | 0 (control) | 24 | hr | 168.24 | 91.00 | p-Akt | 67.96 | ||
Triciribine | T47D | 0 (control) | 24 | hr | 186.87 | 92.32 | p-Akt | 71.34 | ||
Gefitinib | MCF 10A | 0 (control) | 24 | hr | 295.80 | 110.01 | p-Akt | 55.06 | ||
Torkinib | MCF 10A | 0 (control) | 24 | hr | 335.16 | 114.92 | p-Akt | 54.49 | ||
MK2206 | MCF 10A | 0 (control) | 24 | hr | 334.53 | 120.26 | p-Akt | 52.16 | ||
Triciribine | MCF 10A | 0 (control) | 24 | hr | 333.49 | 112.55 | p-Akt | 47.91 | ||
Torkinib | T47D | 0 (control) | 24 | hr | 176.46 | 94.89 | p-Akt | 74.20 | ||
GSK1059615 | AU565 | 0 (control) | 24 | hr | 452.11 | 110.23 | p-Akt | 88.09 | ||
Gefitinib | HCC1954 | 0 (control) | 24 | hr | 342.49 | 120.54 | p-Akt | 84.26 | ||
MK2206 | T47D | 0 (control) | 24 | hr | 176.28 | 99.14 | p-Akt | 70.51 | ||
Torkinib | HCC1954 | 0 (control) | 24 | hr | 309.60 | 109.35 | p-Akt | 76.75 | ||
MK2206 | AU565 | 0 (control) | 24 | hr | 427.04 | 124.23 | p-Akt | 78.88 | ||
GSK1059615 | HCC1954 | 0 (control) | 24 | hr | 302.50 | 106.62 | p-Akt | 73.55 | ||
Torkinib | AU565 | 0 (control) | 24 | hr | 522.19 | 120.45 | p-Akt | 94.97 | ||
MK2206 | HCC1954 | 0 (control) | 24 | hr | 288.09 | 111.00 | p-Akt | 78.02 | ||
Triciribine | AU565 | 0 (control) | 24 | hr | 511.74 | 118.54 | p-Akt | 102.35 | ||
Triciribine | HCC1954 | 0 (control) | 24 | hr | 282.25 | 98.69 | p-Akt | 60.55 | ||
Gefitinib | AU565 | 0 (control) | 24 | hr | 659.08 | 130.41 | p-Akt | 134.35 | ||
Dactolisib | HCC1954 | 0 (control) | 24 | hr | 357.28 | 117.27 | p-Akt | 79.92 | ||
Dactolisib | AU565 | 0 (control) | 24 | hr | 496.14 | 121.03 | p-Akt | 137.91 | ||
Gefitinib | AU565 | 1.0 | nM | 24 | hr | 556.22 | 122.40 | p-Akt | 136.15 |