XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
-6.1
10
uM
XMD8-85 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-12.5
10
uM
XMD8-85 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
3.7
10
uM
XMD8-85 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
-11.6
10
uM
XMD8-85 HeLa SYK
ISDFGLSkALR
Activation Loop
-12.8
10
uM
XMD8-85 HeLa TLK1
YAAVkIHQLNK
Lys1
-38.6
10
uM
XMD8-85 PC-3 TLK1
YAAVkIHQLNK
Lys1
-5.2
10
uM
XMD8-85 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-4.3
10
uM
XMD8-85 HeLa AurB
SHFIVALkVLFK
Lys1
21.7
10
uM
XMD8-85 PC-3 CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
6.2
10
uM
XMD8-85 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
28.6
10
uM
XMD8-85 HeLa MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
-40.4
10
uM
XMD8-85 PC-3 SNRK
DLkPENVVFFEK
Lys2
6.6
10
uM
XMD8-85 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-47.0
10
uM