XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-85 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | -0.3 | 10 | uM |
| XMD8-85 | PC-3 | SRPK1/2 | FVAMkVVK | Lys1 | 11.6 | 10 | uM |
| XMD8-85 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | -13.9 | 10 | uM |
| XMD8-85 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | 21.9 | 10 | uM |
| XMD8-85 | HeLa | KPCI | IYAMkVVK | Lys1 | -10.4 | 10 | uM |
| XMD8-85 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -0.1 | 10 | uM |
| XMD8-85 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -2.3 | 10 | uM |
| XMD8-85 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 49.7 | 10 | uM |
| XMD8-85 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -24.1 | 10 | uM |
| XMD8-85 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | -1.5 | 10 | uM |
| XMD8-85 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | 9.0 | 10 | uM |
| XMD8-85 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | -10.6 | 10 | uM |
| XMD8-85 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | -22.8 | 10 | uM |
| XMD8-85 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | 13.5 | 10 | uM |
| XMD8-85 | HeLa | GCN2 | LDGCCYAVkR | Lys1 | -15.2 | 10 | uM |
| XMD8-85 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | 1.3 | 10 | uM |
| XMD8-85 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | 10.6 | 10 | uM |
| XMD8-85 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -25.7 | 10 | uM |
| XMD8-85 | PC-3 | M4K3 | NVNTGELAAIkVIK | Lys1 | -2.9 | 10 | uM |
| XMD8-85 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | 17.7 | 10 | uM |
| XMD8-85 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | 11.7 | 10 | uM |
| XMD8-85 | PC-3 | MK11 | QELNkTVWEVPQR | Other | 6.3 | 10 | uM |
| XMD8-85 | PC-3 | PDK1 | EYAIkILEK | Lys1 | -22.6 | 10 | uM |
| XMD8-85 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 20.5 | 10 | uM |
| XMD8-85 | HeLa | PKD2 | DVAVkVIDK | Lys1 | -1.2 | 10 | uM |