HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
HG-6-64-01 | A-375 | ABL,ARG | LMTGDTYTAHAGAKFPIK | ACT | 96.2 | 10 | uM |
HG-6-64-01 | A-375 | NEK3 | SKNIFLTQNGK | ACT | 10 | uM | |
HG-6-64-01 | A-375 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | ACT | 74.2 | 10 | uM |
HG-6-64-01 | A-375 | CSK | VSDFGLTKEASSTQDTGKLPVK | ACT | 97.0 | 10 | uM |
HG-6-64-01 | A-375 | RSK2 (Domain 1) | LTDFGLSKESIDHEK | ACT | 17.9 | 10 | uM |
HG-6-64-01 | A-375 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | ACT | 12.0 | 10 | uM |
HG-6-64-01 | A-375 | AXL | KIYNGDYYR | ACT | 10 | uM | |
HG-6-64-01 | A-375 | EPHB4 | FLEENSSDPTYTSSLGGKIPIR | ACT | -1.0 | 10 | uM |
HG-6-64-01 | A-375 | EPHA2 | VLEDDPEATYTTSGGKIPIR | ACT | 66.8 | 10 | uM |
HG-6-64-01 | A-375 | Wnk1,Wnk2,Wnk4 | IGDLGLATLKR | ACT | 0.6 | 10 | uM |
HG-6-64-01 | A-375 | MET | DMYDKEYYSVHNK | ACT | -0.9 | 10 | uM |
HG-6-64-01 | A-375 | eEF2K | YIKYNSNSGFVR | ATP | 26.2 | 10 | uM |
HG-6-64-01 | A-375 | PKCh | VLGKGSFGKVMLAR | ATP | 10 | uM | |
HG-6-64-01 | A-375 | AKT1 | GTFGKVILVK | ATP | 3.8 | 10 | uM |
HG-6-64-01 | A-375 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP | 10 | uM | |
HG-6-64-01 | A-375 | CK1g1/2/3 | KIGCGNFGELR | ATP | 10 | uM | |
HG-6-64-01 | A-375 | COT | GAFGKVYLAQDIK | ATP | 10 | uM | |
HG-6-64-01 | A-375 | PRPK | FLSGLELVKQGAEAR | ATP | 6.3 | 10 | uM |
HG-6-64-01 | A-375 | AurA,AurB,AurC | GKFGNVYLAR | ATP | 9.6 | 10 | uM |
HG-6-64-01 | A-375 | MSK1,MSK2_domain1 | VLGTGAYGKVFLVR | ATP | 28.0 | 10 | uM |
HG-6-64-01 | A-375 | CASK | ETGQQFAVKIVDVAK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | CaMKK2 | LAYNENDNTYYAMKVLSK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | M3K2 | ELAVKQVQFDPDSPETSKEVNALECEIQLLK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | CaMK2g | TSTQEYAAKIINTK | K1 | 2.5 | 10 | uM |
HG-6-64-01 | A-375 | CHK2 | VAIKIISK | K1 | 10 | uM |