HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
HG-6-64-01 | A-375 | NEK7 | AACLLDGVPVALKK | K1 | -26.1 | 10 | uM |
HG-6-64-01 | A-375 | PRP4 | AAGIGKDFKENPNLR | 10.8 | 10 | uM | |
HG-6-64-01 | A-375 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | K2 | 49.4 | 10 | uM |
HG-6-64-01 | A-375 | PIP4K2B | AKDLPTFKDNDFLNEGQK | LIP (PI5K) | -37.8 | 10 | uM |
HG-6-64-01 | A-375 | PIP4K2A | AKELPTLKDNDFINEGQK | LIP (PI5K) | -2.6 | 10 | uM |
HG-6-64-01 | A-375 | LATS1 | ALYATKTLR | K1 | 15.4 | 10 | uM |
HG-6-64-01 | A-375 | MLKL | APVAIKVFK | K1 | -7.5 | 10 | uM |
HG-6-64-01 | A-375 | PHKg2 | ATGHEFAVKIMEVTAER | K1 | 2.7 | 10 | uM |
HG-6-64-01 | A-375 | RSK1 (Domain 2) | ATNMEYAVKVIDK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | AGK | ATVFLNPAACKGK | LIP | ~NI | 10 | uM |
HG-6-64-01 | A-375 | PLK1 like (splice variant or novel kinase) | CFEISDADNKVVFAGKIVPK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PLK1 | CFEISDADTKEVFAGKIVPK | K1 | 3.4 | 10 | uM |
HG-6-64-01 | A-375 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIKTCK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | CDK8 | DGKDDKDYALKQIEGTGISMSACR | K1 | 10 | uM | |
HG-6-64-01 | A-375 | MST3 | DIKAANVLLSEHGEVK | K2 | -5.1 | 10 | uM |
HG-6-64-01 | A-375 | MST4,YSK1 | DIKAANVLLSEQGDVK | K2 | -26.0 | 10 | uM |
HG-6-64-01 | A-375 | MST1,MST2 | DIKAGNILLNTEGHAK | K2 | 18.3 | 10 | uM |
HG-6-64-01 | A-375 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | K2 | ND | 10 | uM |
HG-6-64-01 | A-375 | CDK13 | DIKCSNILLNNRGQIK | K2 | 14.2 | 10 | uM |
HG-6-64-01 | A-375 | CRK7 | DIKCSNILLNNSGQIK | K2 | 10 | uM | |
HG-6-64-01 | A-375 | MAP3K4 | DIKGANIFLTSSGLIK | K2 | -21.8 | 10 | uM |
HG-6-64-01 | A-375 | KHS1 | DIKGANILLTDHGDVK | K2 | 35.0 | 10 | uM |
HG-6-64-01 | A-375 | M3K2,MAP3K3 | DIKGANILR | K2 | 11.7 | 10 | uM |
HG-6-64-01 | A-375 | GCK | DIKGANLLLTLQGDVK | K2 | 10 | uM | |
HG-6-64-01 | A-375 | MAP3K5 | DIKGDNVLINTYSGVLK | K2 | -9.4 | 10 | uM |