HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| HG-6-64-01 | A-375 | MK14 | QELNKTIWEVPER | Other (MAPKAP2/3 active site in p38a complex) | 97.3 | 10 | uM |
| HG-6-64-01 | A-375 | CHK1 | LSKGDGLEFK | nonKD (autoinhibition domain) | 30.0 | 10 | uM |
| HG-6-64-01 | A-375 | PIK4CB | VPHTQAVVLNSKDKAPYLIYVEVLECENFDTTSVPARIPENR | nonKD | -58.2 | 10 | uM |
| HG-6-64-01 | A-375 | PIP4K2A | AKELPTLKDNDFINEGQK | LIP (PI5K) | -2.6 | 10 | uM |
| HG-6-64-01 | A-375 | FYV1 | GGKSGAAFYATEDDRFILK | LIP (PI5K) | -22.6 | 10 | uM |
| HG-6-64-01 | A-375 | PIP4K2B | AKDLPTFKDNDFLNEGQK | LIP (PI5K) | -37.8 | 10 | uM |
| HG-6-64-01 | A-375 | PI42C | VKELPTLKDMDFLNK | LIP (PI5K) | -4.7 | 10 | uM |
| HG-6-64-01 | A-375 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | LIP (PI5K) | 9.6 | 10 | uM |
| HG-6-64-01 | A-375 | PIK3C2B | VIFKCGDDLRQDMLTLQMIR | LIP (PI3K/PI4K) | 16.5 | 10 | uM |
| HG-6-64-01 | A-375 | PIK3CB | VFGEDSVGVIFKNGDDLRQDMLTLQMLR | LIP (PI3K/PI4K) | 10 | uM | |
| HG-6-64-01 | A-375 | PIK3C3 | TEDGGKYPVIFKHGDDLR | LIP (PI3K/PI4K) | 16.3 | 10 | uM |
| HG-6-64-01 | A-375 | ATM | QLVKGRDDLRQDAVMQQVFQMCNTLLQR | LIP | 10 | uM | |
| HG-6-64-01 | A-375 | AGK | ATVFLNPAACKGK | LIP | ~NI | 10 | uM |
| HG-6-64-01 | A-375 | FRAP1 | IQSIAPSLQVITSKQRPR | LIP | ~NI | 10 | uM |
| HG-6-64-01 | A-375 | SMG1 | DTVTIHSVGGTITILPTKTKPK | LIP | 12.2 | 10 | uM |
| HG-6-64-01 | A-375 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | LIP | 13.7 | 10 | uM |
| HG-6-64-01 | A-375 | ATR | FYIMMCKPK | LIP | 9.7 | 10 | uM |
| HG-6-64-01 | A-375 | ULK2 | NLSKSQILLGKEIKILK | KD | 10 | uM | |
| HG-6-64-01 | A-375 | CK2a2 | LIDTVKDPVSK | KD | 10 | uM | |
| HG-6-64-01 | A-375 | PAN3 | VMDPTKILITGK | KD | 10 | uM | |
| HG-6-64-01 | A-375 | IKKE,TBK1 | DIKPGNIMR | K2 | 10 | uM | |
| HG-6-64-01 | A-375 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | K2 | 49.4 | 10 | uM |
| HG-6-64-01 | A-375 | GSK3B | DIKPQNLLLDPDTAVLK | K2 | 15.2 | 10 | uM |
| HG-6-64-01 | A-375 | MK03 | DLKPSNLLINTTCDLK | K2 | 0.9 | 10 | uM |
| HG-6-64-01 | A-375 | IKKA | DLKPENIVLQDVGGK | K2 | 38.5 | 10 | uM |