HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
HG-6-64-01 A-375 ZC3 (MINK)
TGQLAAIKVMDVTEDEEEEIKQEINMLKK
K1
10
uM
HG-6-64-01 A-375 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIKGQNVLLTENAEVK
K2
60.3
10
uM
HG-6-64-01 A-375 Wnk1,Wnk2,Wnk4
IGDLGLATLKR
ACT
0.6
10
uM
HG-6-64-01 A-375 Wnk1,Wnk2,Wnk3
DLKCDNIFITGPTGSVK
K2
-12.9
10
uM
HG-6-64-01 A-375 WEE1
YIHSMSLVHMDIKPSNIFISR
K2
13.1
10
uM
HG-6-64-01 A-375 ULK3
NISHLDLKPQNILLSSLEKPHLK
K2
-7.7
10
uM
HG-6-64-01 A-375 ULK2
NLSKSQILLGKEIKILK
KD
10
uM
HG-6-64-01 A-375 TNK1
SVPVAVKSLR
K1
10
uM
HG-6-64-01 A-375 TLK1/2
YLNEIKPPIIHYDLKPGNILLVNGTACGEIK
K2
10
uM
HG-6-64-01 A-375 TLK1
YLNEIKPPIIHYDLKPGNILLVDGTACGEIK
K2
10
uM
HG-6-64-01 A-375 TIF1b
VLVNDAQKVTEGQQER
~NI
10
uM
HG-6-64-01 A-375 TIF1b
QGSGSSQPMEVQEGYGFGSGDDPYSSAEPHVSGVKR
ND
10
uM
HG-6-64-01 A-375 TAOK2
DVKAGNILLSEPGLVK
K2
21.1
10
uM
HG-6-64-01 A-375 TAO1,TAOK3
DIKAGNILLTEPGQVK
K2
ND
10
uM
HG-6-64-01 A-375 STLK6
HTPTGTLVTIKITNLENCNEER
10
uM
HG-6-64-01 A-375 SRPK1/2
FVAMKVVK
K1
10
uM
HG-6-64-01 A-375 SRPK1
IIHTDIKPENILLSVNEQYIR
K2
6.7
10
uM
HG-6-64-01 A-375 SMG1
DTVTIHSVGGTITILPTKTKPK
LIP
12.2
10
uM
HG-6-64-01 A-375 SLK
DLKAGNILFTLDGDIK
-1.1
10
uM
HG-6-64-01 A-375 SIK3
VAIKIIDKTQLDEENLK
K1
10
uM
HG-6-64-01 A-375 SGK3
DLKPENILLDSVGHVVLTDFGLCK
K2
ND
10
uM
HG-6-64-01 A-375 SGK3
FYAVKVLQK
K1
6.8
10
uM
HG-6-64-01 A-375 SGK1
HKAEEVFYAVKVLQKK
K1
10
uM
HG-6-64-01 A-375 RSK2_domain2
DLKPSNILYVDESGNPESIR
K2
4.3
10
uM
HG-6-64-01 A-375 RSK2 (Domain 1)
LTDFGLSKESIDHEK
ACT
17.9
10
uM
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