HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
HG-6-64-01 | A-375 | ZC3 (MINK) | TGQLAAIKVMDVTEDEEEEIKQEINMLKK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | K2 | 60.3 | 10 | uM |
HG-6-64-01 | A-375 | Wnk1,Wnk2,Wnk4 | IGDLGLATLKR | ACT | 0.6 | 10 | uM |
HG-6-64-01 | A-375 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | K2 | -12.9 | 10 | uM |
HG-6-64-01 | A-375 | WEE1 | YIHSMSLVHMDIKPSNIFISR | K2 | 13.1 | 10 | uM |
HG-6-64-01 | A-375 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | K2 | -7.7 | 10 | uM |
HG-6-64-01 | A-375 | ULK2 | NLSKSQILLGKEIKILK | KD | 10 | uM | |
HG-6-64-01 | A-375 | TNK1 | SVPVAVKSLR | K1 | 10 | uM | |
HG-6-64-01 | A-375 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | K2 | 10 | uM | |
HG-6-64-01 | A-375 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | K2 | 10 | uM | |
HG-6-64-01 | A-375 | TIF1b | VLVNDAQKVTEGQQER | ~NI | 10 | uM | |
HG-6-64-01 | A-375 | TIF1b | QGSGSSQPMEVQEGYGFGSGDDPYSSAEPHVSGVKR | ND | 10 | uM | |
HG-6-64-01 | A-375 | TAOK2 | DVKAGNILLSEPGLVK | K2 | 21.1 | 10 | uM |
HG-6-64-01 | A-375 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | K2 | ND | 10 | uM |
HG-6-64-01 | A-375 | STLK6 | HTPTGTLVTIKITNLENCNEER | 10 | uM | ||
HG-6-64-01 | A-375 | SRPK1/2 | FVAMKVVK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | SRPK1 | IIHTDIKPENILLSVNEQYIR | K2 | 6.7 | 10 | uM |
HG-6-64-01 | A-375 | SMG1 | DTVTIHSVGGTITILPTKTKPK | LIP | 12.2 | 10 | uM |
HG-6-64-01 | A-375 | SLK | DLKAGNILFTLDGDIK | -1.1 | 10 | uM | |
HG-6-64-01 | A-375 | SIK3 | VAIKIIDKTQLDEENLK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | SGK3 | DLKPENILLDSVGHVVLTDFGLCK | K2 | ND | 10 | uM |
HG-6-64-01 | A-375 | SGK3 | FYAVKVLQK | K1 | 6.8 | 10 | uM |
HG-6-64-01 | A-375 | SGK1 | HKAEEVFYAVKVLQKK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | K2 | 4.3 | 10 | uM |
HG-6-64-01 | A-375 | RSK2 (Domain 1) | LTDFGLSKESIDHEK | ACT | 17.9 | 10 | uM |