Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
BT-20 | Palbociclib | 0.1 | CDK4/6 | Cell cycle | 0.3557 | 0.03619 |
BT-20 | Palbociclib | 0.31623 | CDK4/6 | Cell cycle | 0.2359 | 0.04751 |
BT-20 | Palbociclib | 1.0 | CDK4/6 | Cell cycle | 0.2044 | 0.04646 |
BT-20 | Palbociclib | 3.1623 | CDK4/6 | Cell cycle | 0.1624 | 0.05010 |
BT-20 | AZD7762 | 0.001 | CHK1/2 | Cell cycle | 1.1198 | -0.00253 |
BT-20 | AZD7762 | 0.0031623 | CHK1/2 | Cell cycle | 1.2431 | -0.00726 |
BT-20 | AZD7762 | 0.01 | CHK1/2 | Cell cycle | 1.2200 | 0.00225 |
BT-20 | AZD7762 | 0.031623 | CHK1/2 | Cell cycle | 1.2229 | 0.01175 |
BT-20 | AZD7762 | 0.1 | CHK1/2 | Cell cycle | 1.1714 | 0.04490 |
BT-20 | AZD7762 | 0.31623 | CHK1/2 | Cell cycle | 0.9454 | 0.07692 |
BT-20 | AZD7762 | 1.0 | CHK1/2 | Cell cycle | 0.5068 | 0.21188 |
BT-20 | AZD7762 | 3.1623 | CHK1/2 | Cell cycle | -0.1525 | 0.50057 |
BT-20 | AZD7762 | 10.0 | CHK1/2 | Cell cycle | -0.5785 | 0.71162 |
BT-20 | Volasertib | 0.0001 | PLK | Cell cycle | 1.0476 | -0.00114 |
BT-20 | Volasertib | 0.00031623 | PLK | Cell cycle | 1.0308 | 0.00572 |
BT-20 | Volasertib | 0.001 | PLK | Cell cycle | 1.0085 | 0.00742 |
BT-20 | Volasertib | 0.0031623 | PLK | Cell cycle | 0.8266 | 0.05236 |
BT-20 | Volasertib | 0.01 | PLK | Cell cycle | 0.0133 | 0.34529 |
BT-20 | Volasertib | 0.031623 | PLK | Cell cycle | -0.4356 | 0.63889 |
BT-20 | Volasertib | 0.1 | PLK | Cell cycle | -0.5218 | 0.70449 |
BT-20 | Volasertib | 0.31623 | PLK | Cell cycle | -0.5339 | 0.71936 |
BT-20 | Volasertib | 1.0 | PLK | Cell cycle | -0.4694 | 0.64260 |
BT-20 | Dinaciclib | 0.0001 | pan CDK | Cell cycle | 0.9253 | 0.00567 |
BT-20 | Dinaciclib | 0.00031623 | pan CDK | Cell cycle | 1.0258 | -0.00375 |
BT-20 | Dinaciclib | 0.001 | pan CDK | Cell cycle | 1.0071 | -0.00417 |