Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)

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Cell Small Molecule Small Mol Concentration (uM) Primary Target Pathway Mean Normalized Growth Rate Inhibition Value Increased Fraction Dead
BT-20 Palbociclib
0.1
CDK4/6
Cell cycle
0.3557 0.03619
BT-20 Palbociclib
0.31623
CDK4/6
Cell cycle
0.2359 0.04751
BT-20 Palbociclib
1.0
CDK4/6
Cell cycle
0.2044 0.04646
BT-20 Palbociclib
3.1623
CDK4/6
Cell cycle
0.1624 0.05010
BT-20 AZD7762
0.001
CHK1/2
Cell cycle
1.1198 -0.00253
BT-20 AZD7762
0.0031623
CHK1/2
Cell cycle
1.2431 -0.00726
BT-20 AZD7762
0.01
CHK1/2
Cell cycle
1.2200 0.00225
BT-20 AZD7762
0.031623
CHK1/2
Cell cycle
1.2229 0.01175
BT-20 AZD7762
0.1
CHK1/2
Cell cycle
1.1714 0.04490
BT-20 AZD7762
0.31623
CHK1/2
Cell cycle
0.9454 0.07692
BT-20 AZD7762
1.0
CHK1/2
Cell cycle
0.5068 0.21188
BT-20 AZD7762
3.1623
CHK1/2
Cell cycle
-0.1525 0.50057
BT-20 AZD7762
10.0
CHK1/2
Cell cycle
-0.5785 0.71162
BT-20 Volasertib
0.0001
PLK
Cell cycle
1.0476 -0.00114
BT-20 Volasertib
0.00031623
PLK
Cell cycle
1.0308 0.00572
BT-20 Volasertib
0.001
PLK
Cell cycle
1.0085 0.00742
BT-20 Volasertib
0.0031623
PLK
Cell cycle
0.8266 0.05236
BT-20 Volasertib
0.01
PLK
Cell cycle
0.0133 0.34529
BT-20 Volasertib
0.031623
PLK
Cell cycle
-0.4356 0.63889
BT-20 Volasertib
0.1
PLK
Cell cycle
-0.5218 0.70449
BT-20 Volasertib
0.31623
PLK
Cell cycle
-0.5339 0.71936
BT-20 Volasertib
1.0
PLK
Cell cycle
-0.4694 0.64260
BT-20 Dinaciclib
0.0001
pan CDK
Cell cycle
0.9253 0.00567
BT-20 Dinaciclib
0.00031623
pan CDK
Cell cycle
1.0258 -0.00375
BT-20 Dinaciclib
0.001
pan CDK
Cell cycle
1.0071 -0.00417