Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
BT-20 | A-1210477 | 0.0031623 | Mcl-1 | Misc | 0.9994 | -0.00302 |
BT-20 | A-1210477 | 0.01 | Mcl-1 | Misc | 1.0461 | 0.00227 |
BT-20 | A-1210477 | 0.31623 | Mcl-1 | Misc | 1.0544 | -0.00191 |
BT-20 | A-1210477 | 1.0 | Mcl-1 | Misc | 1.0474 | -0.00138 |
BT-20 | A-1210477 | 10.0 | Mcl-1 | Misc | 0.8209 | 0.04589 |
BT-20 | Olaparib | 0.001 | PARP | Misc | 1.0265 | -0.00519 |
BT-20 | Olaparib | 0.31623 | PARP | Misc | 0.9400 | 0.00840 |
BT-20 | Olaparib | 1.0 | PARP | Misc | 0.9125 | 0.00565 |
BT-20 | Olaparib | 10.0 | PARP | Misc | 0.6064 | 0.04246 |
BT-20 | Bleomycin | 0.0010833 | Radiation | Misc | 0.9824 | 0.00530 |
BT-20 | Bleomycin | 0.031667 | Radiation | Misc | 0.9548 | 0.00025 |
BT-20 | Bleomycin | 0.1 | Radiation | Misc | 0.8145 | 0.02731 |
BT-20 | Bleomycin | 1.0 | Radiation | Misc | 0.3200 | 0.15033 |
BT-20 | Bleomycin | 3.1623 | Radiation | Misc | -0.0603 | 0.30083 |
BT-20 | Ipatasertib | 0.01 | AKT | PI3K/mTOR | 0.9717 | -0.00176 |
BT-20 | Ipatasertib | 0.031623 | AKT | PI3K/mTOR | 0.9656 | 0.00133 |
BT-20 | Ipatasertib | 0.31623 | AKT | PI3K/mTOR | 0.5886 | 0.02673 |
BT-20 | Ipatasertib | 1.0 | AKT | PI3K/mTOR | 0.4168 | 0.05632 |
BT-20 | Alpelisib | 0.001 | PI3Ka | PI3K/mTOR | 1.0513 | 0.00412 |
BT-20 | Alpelisib | 0.0031623 | PI3Ka | PI3K/mTOR | 1.0511 | 0.01061 |
BT-20 | Alpelisib | 0.031623 | PI3Ka | PI3K/mTOR | 0.9920 | 0.01246 |
BT-20 | Alpelisib | 0.1 | PI3Ka | PI3K/mTOR | 0.9578 | 0.00889 |
BT-20 | Taselisib | 0.0031623 | PI3Ka, g, d | PI3K/mTOR | 0.8758 | 0.02377 |
BT-20 | Everolimus | 10.0 | mTOR1 | PI3K/mTOR | 0.3900 | 0.07549 |
BT-20 | Everolimus | 3.1623 | mTOR1 | PI3K/mTOR | 0.4209 | 0.06403 |