Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
T47D | AZD7762 | 0.01 | CHK1/2 | Cell cycle | 1.3830 | -0.00136 |
PDXHCI002 | Torin2 | 0.0031623 | mTOR/ATM/ATR | PI3K/mTOR | 1.3716 | -0.03537 |
HCC70 | AZD7762 | 0.0031623 | CHK1/2 | Cell cycle | 1.3706 | -0.00299 |
MDA-MB-134-VI | Cabozantinib | 1.0 | VEGFR2/MET | RTK | 1.3646 | -0.00006 |
MDA-MB-134-VI | Neratinib | 0.001 | EGFR/HER2 | RTK | 1.3618 | -0.00624 |
CAL-85-1 | AZD7762 | 0.0031623 | CHK1/2 | Cell cycle | 1.3608 | -0.00028 |
MDA-MB-134-VI | Cabozantinib | 0.001 | VEGFR2/MET | RTK | 1.3562 | -0.00502 |
MDA-MB-134-VI | Luminespib | 0.0001 | HSP90 | Misc | 1.3453 | -0.00808 |
MDA-MB-134-VI | PF-4708671 | 0.01 | p70S6K | PI3K/mTOR | 1.3419 | -0.00121 |
HCC1419 | Volasertib | 0.00031623 | PLK | Cell cycle | 1.3365 | 0.00331 |
MDA-MB-134-VI | Luminespib | 0.00031623 | HSP90 | Misc | 1.3361 | -0.01039 |
MDA-MB-134-VI | Neratinib | 0.00031623 | EGFR/HER2 | RTK | 1.3354 | 0.00352 |
PDXHCI002 | INK-128 | 0.01 | mTORC1/2 | PI3K/mTOR | 1.3353 | -0.05354 |
MDA-MB-134-VI | Cediranib | 0.0031623 | VEGFR/cKIT | RTK | 1.3300 | -0.00799 |
MDA-MB-134-VI | Vorinostat | 0.31623 | HDAC | Misc | 1.3286 | 0.00076 |
HCC70 | Abemaciclib | 0.0031623 | CDK4/6 | Cell cycle | 1.3213 | -0.01140 |
MDA-MB-134-VI | Cediranib | 1.0 | VEGFR/cKIT | RTK | 1.3176 | 0.01247 |
MDA-MB-134-VI | Alpelisib | 0.0031623 | PI3Ka | PI3K/mTOR | 1.3174 | -0.00250 |
MDA-MB-134-VI | Cediranib | 0.001 | VEGFR/cKIT | RTK | 1.3158 | -0.01192 |
HCC1419 | Vorinostat | 0.31623 | HDAC | Misc | 1.3152 | -0.00210 |
HCC70 | Volasertib | 0.00031623 | PLK | Cell cycle | 1.3093 | 0.00186 |
MDA-MB-453 | Vorinostat | 0.31623 | HDAC | Misc | 1.3002 | 0.00416 |
HCC1500 | Etoposide | 0.031667 | Topo II | Chemotherapy | 1.2999 | -0.03422 |
MDA-MB-453 | Ipatasertib | 0.01 | AKT | PI3K/mTOR | 1.2982 | -0.02244 |
T47D | AZD7762 | 0.1 | CHK1/2 | Cell cycle | 1.2980 | 0.00257 |