Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
T47D | Ipatasertib | 0.31623 | AKT | PI3K/mTOR | 0.3286 | 0.01648 |
T47D | Ipatasertib | 1.0 | AKT | PI3K/mTOR | 0.1884 | 0.01828 |
T47D | Ipatasertib | 3.1623 | AKT | PI3K/mTOR | 0.1331 | 0.02540 |
T47D | Ipatasertib | 10.0 | AKT | PI3K/mTOR | 0.1402 | 0.02929 |
T47D | Alpelisib | 0.001 | PI3Ka | PI3K/mTOR | 1.0781 | 0.00072 |
T47D | Alpelisib | 0.0031623 | PI3Ka | PI3K/mTOR | 1.0415 | 0.00157 |
T47D | Alpelisib | 0.01 | PI3Ka | PI3K/mTOR | 0.8915 | 0.00055 |
T47D | Alpelisib | 0.031623 | PI3Ka | PI3K/mTOR | 0.7429 | 0.00918 |
T47D | Alpelisib | 0.1 | PI3Ka | PI3K/mTOR | 0.5767 | 0.00912 |
T47D | Alpelisib | 0.31623 | PI3Ka | PI3K/mTOR | 0.3518 | 0.01207 |
T47D | Alpelisib | 1.0 | PI3Ka | PI3K/mTOR | 0.1904 | 0.02302 |
T47D | Alpelisib | 3.1623 | PI3Ka | PI3K/mTOR | 0.0422 | 0.03677 |
T47D | Alpelisib | 10.0 | PI3Ka | PI3K/mTOR | -0.0332 | 0.06965 |
T47D | Taselisib | 0.001 | PI3Ka, g, d | PI3K/mTOR | 0.6727 | 0.00360 |
T47D | Taselisib | 0.0031623 | PI3Ka, g, d | PI3K/mTOR | 0.3265 | 0.02050 |
T47D | Taselisib | 0.01 | PI3Ka, g, d | PI3K/mTOR | 0.1037 | 0.03585 |
T47D | Taselisib | 0.031623 | PI3Ka, g, d | PI3K/mTOR | 0.0519 | 0.04296 |
T47D | Taselisib | 0.1 | PI3Ka, g, d | PI3K/mTOR | 0.0051 | 0.04903 |
T47D | Taselisib | 0.31623 | PI3Ka, g, d | PI3K/mTOR | -0.0046 | 0.06924 |
T47D | Taselisib | 1.0 | PI3Ka, g, d | PI3K/mTOR | 0.0382 | 0.06275 |
T47D | Taselisib | 3.1623 | PI3Ka, g, d | PI3K/mTOR | 0.0034 | 0.07274 |
T47D | Taselisib | 10.0 | PI3Ka, g, d | PI3K/mTOR | -0.1047 | 0.13876 |
T47D | TGX221 | 0.001 | PI3Kb | PI3K/mTOR | 1.0725 | 0.00126 |
T47D | TGX221 | 0.0031623 | PI3Kb | PI3K/mTOR | 1.0733 | -0.00116 |
T47D | TGX221 | 0.01 | PI3Kb | PI3K/mTOR | 1.0730 | 0.00055 |