AS-252424 KINOMEscan - Dataset (ID:20341)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
AS-252424 | IGF1R | 100.0 | 10000 | nM |
AS-252424 | IKKA | 47.7 | 10000 | nM |
AS-252424 | IKKB | 100.0 | 10000 | nM |
AS-252424 | IKKE | 100.0 | 10000 | nM |
AS-252424 | INSR | 95.9 | 10000 | nM |
AS-252424 | INSRR | 55.9 | 10000 | nM |
AS-252424 | IRAK3 | 78.0 | 10000 | nM |
AS-252424 | ITK | 100.0 | 10000 | nM |
AS-252424 | JAK1(JH1domain-catalytic) | 100.0 | 10000 | nM |
AS-252424 | JAK1(JH2domain-pseudokinase) | 51.1 | 10000 | nM |
AS-252424 | JAK2(JH1domain-catalytic) | 100.0 | 10000 | nM |
AS-252424 | JAK3(JH1domain-catalytic) | 85.1 | 10000 | nM |
AS-252424 | JNK1 | 100.0 | 10000 | nM |
AS-252424 | MK09 | 79.7 | 10000 | nM |
AS-252424 | JNK3 | 38.1 | 10000 | nM |
AS-252424 | KIT | 100.0 | 10000 | nM |
AS-252424 | KIT(D816V) | 100.0 | 10000 | nM |
AS-252424 | KIT(V559D) | 87.1 | 10000 | nM |
AS-252424 | KIT(V559D,T670I) | 80.6 | 10000 | nM |
AS-252424 | KIT(V559D,V654A) | 84.2 | 10000 | nM |
AS-252424 | LATS1 | 100.0 | 10000 | nM |
AS-252424 | LATS2 | 100.0 | 10000 | nM |
AS-252424 | LCK | 77.2 | 10000 | nM |
AS-252424 | LIMK1 | 100.0 | 10000 | nM |
AS-252424 | LIMK2 | 81.9 | 10000 | nM |