AS-252424 KINOMEscan - Dataset (ID:20341)

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Small Molecule Protein % Control Assay compound conc Conc unit
AS-252424 IGF1R 100.0 10000
nM
AS-252424 IKKA 47.7 10000
nM
AS-252424 IKKB 100.0 10000
nM
AS-252424 IKKE 100.0 10000
nM
AS-252424 INSR 95.9 10000
nM
AS-252424 INSRR 55.9 10000
nM
AS-252424 IRAK3 78.0 10000
nM
AS-252424 ITK 100.0 10000
nM
AS-252424 JAK1(JH1domain-catalytic) 100.0 10000
nM
AS-252424 JAK1(JH2domain-pseudokinase) 51.1 10000
nM
AS-252424 JAK2(JH1domain-catalytic) 100.0 10000
nM
AS-252424 JAK3(JH1domain-catalytic) 85.1 10000
nM
AS-252424 JNK1 100.0 10000
nM
AS-252424 MK09 79.7 10000
nM
AS-252424 JNK3 38.1 10000
nM
AS-252424 KIT 100.0 10000
nM
AS-252424 KIT(D816V) 100.0 10000
nM
AS-252424 KIT(V559D) 87.1 10000
nM
AS-252424 KIT(V559D,T670I) 80.6 10000
nM
AS-252424 KIT(V559D,V654A) 84.2 10000
nM
AS-252424 LATS1 100.0 10000
nM
AS-252424 LATS2 100.0 10000
nM
AS-252424 LCK 77.2 10000
nM
AS-252424 LIMK1 100.0 10000
nM
AS-252424 LIMK2 81.9 10000
nM