AS-252424 KINOMEscan - Dataset (ID:20341)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
AS-252424 | FER | 95.5 | 10000 | nM |
AS-252424 | FES | 100.0 | 10000 | nM |
AS-252424 | FGFR1 | 100.0 | 10000 | nM |
AS-252424 | FGFR2 | 100.0 | 10000 | nM |
AS-252424 | FGFR3 | 100.0 | 10000 | nM |
AS-252424 | FGFR3(G697C) | 92.3 | 10000 | nM |
AS-252424 | FGFR4 | 68.0 | 10000 | nM |
AS-252424 | FGR | 100.0 | 10000 | nM |
AS-252424 | VGFR1 | 68.7 | 10000 | nM |
AS-252424 | FLT3 | 100.0 | 10000 | nM |
AS-252424 | FLT3(D835H) | 88.4 | 10000 | nM |
AS-252424 | FLT3(D835Y) | 100.0 | 10000 | nM |
AS-252424 | FLT3(ITD) | 91.2 | 10000 | nM |
AS-252424 | FLT3(K663Q) | 96.2 | 10000 | nM |
AS-252424 | FLT3(N841I) | 82.3 | 10000 | nM |
AS-252424 | FLT4 | 96.5 | 10000 | nM |
AS-252424 | FRK | 90.9 | 10000 | nM |
AS-252424 | FYN | 88.6 | 10000 | nM |
AS-252424 | GAK | 9.3 | 10000 | nM |
AS-252424 | GCN2(Kin.Dom.2,S808G) | 76.5 | 10000 | nM |
AS-252424 | GSK3A | 64.9 | 10000 | nM |
AS-252424 | GSK3B | 92.4 | 10000 | nM |
AS-252424 | HCK | 100.0 | 10000 | nM |
AS-252424 | HIPK1 | 5.0 | 10000 | nM |
AS-252424 | M4K1 | 95.4 | 10000 | nM |