AS-252424 KINOMEscan - Dataset (ID:20341)

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Small Molecule Protein % Control Assay compound conc Conc unit
AS-252424 FER 95.5 10000
nM
AS-252424 FES 100.0 10000
nM
AS-252424 FGFR1 100.0 10000
nM
AS-252424 FGFR2 100.0 10000
nM
AS-252424 FGFR3 100.0 10000
nM
AS-252424 FGFR3(G697C) 92.3 10000
nM
AS-252424 FGFR4 68.0 10000
nM
AS-252424 FGR 100.0 10000
nM
AS-252424 VGFR1 68.7 10000
nM
AS-252424 FLT3 100.0 10000
nM
AS-252424 FLT3(D835H) 88.4 10000
nM
AS-252424 FLT3(D835Y) 100.0 10000
nM
AS-252424 FLT3(ITD) 91.2 10000
nM
AS-252424 FLT3(K663Q) 96.2 10000
nM
AS-252424 FLT3(N841I) 82.3 10000
nM
AS-252424 FLT4 96.5 10000
nM
AS-252424 FRK 90.9 10000
nM
AS-252424 FYN 88.6 10000
nM
AS-252424 GAK 9.3 10000
nM
AS-252424 GCN2(Kin.Dom.2,S808G) 76.5 10000
nM
AS-252424 GSK3A 64.9 10000
nM
AS-252424 GSK3B 92.4 10000
nM
AS-252424 HCK 100.0 10000
nM
AS-252424 HIPK1 5.0 10000
nM
AS-252424 M4K1 95.4 10000
nM