AS-252424 KINOMEscan - Dataset (ID:20341)

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Small Molecule Protein % Control Assay compound conc Conc unit
AS-252424 EGFR(L747-T751del,Sins) 1.9 10000
nM
AS-252424 EGFR(L858R) 20.1 10000
nM
AS-252424 EGFR(L861Q) 27.6 10000
nM
AS-252424 EGFR(S752-I759del) 9.9 10000
nM
AS-252424 EPHA1 100.0 10000
nM
AS-252424 EPHA2 100.0 10000
nM
AS-252424 EPHA3 100.0 10000
nM
AS-252424 EPHA4 93.1 10000
nM
AS-252424 EPHA5 100.0 10000
nM
AS-252424 EPHA6 92.3 10000
nM
AS-252424 EPHA7 100.0 10000
nM
AS-252424 EPHA8 100.0 10000
nM
AS-252424 EPHB1 100.0 10000
nM
AS-252424 EPHB2 74.6 10000
nM
AS-252424 EPHB3 75.4 10000
nM
AS-252424 EPHB4 100.0 10000
nM
AS-252424 ERBB2 100.0 10000
nM
AS-252424 ERBB4 49.5 10000
nM
AS-252424 MK03 100.0 10000
nM
AS-252424 MK01 100.0 10000
nM
AS-252424 ERK3 80.2 10000
nM
AS-252424 ERK4 100.0 10000
nM
AS-252424 ERK5 100.0 10000
nM
AS-252424 ERK8 3.7 10000
nM
AS-252424 FAK1 100.0 10000
nM