AS-252424 KINOMEscan - Dataset (ID:20341)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
AS-252424 | EGFR(L747-T751del,Sins) | 1.9 | 10000 | nM |
AS-252424 | EGFR(L858R) | 20.1 | 10000 | nM |
AS-252424 | EGFR(L861Q) | 27.6 | 10000 | nM |
AS-252424 | EGFR(S752-I759del) | 9.9 | 10000 | nM |
AS-252424 | EPHA1 | 100.0 | 10000 | nM |
AS-252424 | EPHA2 | 100.0 | 10000 | nM |
AS-252424 | EPHA3 | 100.0 | 10000 | nM |
AS-252424 | EPHA4 | 93.1 | 10000 | nM |
AS-252424 | EPHA5 | 100.0 | 10000 | nM |
AS-252424 | EPHA6 | 92.3 | 10000 | nM |
AS-252424 | EPHA7 | 100.0 | 10000 | nM |
AS-252424 | EPHA8 | 100.0 | 10000 | nM |
AS-252424 | EPHB1 | 100.0 | 10000 | nM |
AS-252424 | EPHB2 | 74.6 | 10000 | nM |
AS-252424 | EPHB3 | 75.4 | 10000 | nM |
AS-252424 | EPHB4 | 100.0 | 10000 | nM |
AS-252424 | ERBB2 | 100.0 | 10000 | nM |
AS-252424 | ERBB4 | 49.5 | 10000 | nM |
AS-252424 | MK03 | 100.0 | 10000 | nM |
AS-252424 | MK01 | 100.0 | 10000 | nM |
AS-252424 | ERK3 | 80.2 | 10000 | nM |
AS-252424 | ERK4 | 100.0 | 10000 | nM |
AS-252424 | ERK5 | 100.0 | 10000 | nM |
AS-252424 | ERK8 | 3.7 | 10000 | nM |
AS-252424 | FAK1 | 100.0 | 10000 | nM |