Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
WM-115 Vemurafenib Vorinostat 1.0000 0.1067
uM
48
hr
1 1612 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 133.39 NGFR rabbit IgG(H+L) / donkey NGFR 1125.00
WM115-B2-rep1
D2
WM-115 Vemurafenib JW55 1.0000 0.1067
uM
48
hr
1 1525 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 145.03 NGFR rabbit IgG(H+L) / donkey NGFR 1076.22
WM115-B2-rep1
D3
WM-115 Vemurafenib Entinostat 1.0000 0.1067
uM
48
hr
1 1701 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 130.88 NGFR rabbit IgG(H+L) / donkey NGFR 1358.88
WM115-B2-rep1
D4
WM-115 Vemurafenib AGK2 1.0000 0.1067
uM
48
hr
1 1420 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 139.59 NGFR rabbit IgG(H+L) / donkey NGFR 1264.14
WM115-B2-rep1
D5
WM-115 Vemurafenib GSK-J4 1.0000 0.1067
uM
48
hr
1 1589 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 141.26 NGFR rabbit IgG(H+L) / donkey NGFR 1214.14
WM115-B2-rep1
D6
WM-115 Vemurafenib (-)-JQ1 1.0000 0.1067
uM
48
hr
1 1461 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 134.05 NGFR rabbit IgG(H+L) / donkey NGFR 1153.67
WM115-B2-rep1
D7
WM-115 Vemurafenib IOX2 1.0000 0.1067
uM
48
hr
1 1508 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 141.26 NGFR rabbit IgG(H+L) / donkey NGFR 1073.48
WM115-B2-rep1
D8
WM-115 Vemurafenib Azacitidine 1.0000 0.1067
uM
48
hr
1 1371 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 156.64 NGFR rabbit IgG(H+L) / donkey NGFR 985.52
WM115-B2-rep1
E2
WM-115 Vemurafenib C646 1.0000 0.1067
uM
48
hr
1 1389 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 144.13 NGFR rabbit IgG(H+L) / donkey NGFR 1023.21
WM115-B2-rep1
E3
WM-115 Vemurafenib Mocetinostat 1.0000 0.1067
uM
48
hr
1 1586 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 123.99 NGFR rabbit IgG(H+L) / donkey NGFR 1412.07
WM115-B2-rep1
E4
WM-115 Vemurafenib Resveratrol 1.0000 0.1067
uM
48
hr
1 1377 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 140.59 NGFR rabbit IgG(H+L) / donkey NGFR 1187.81
WM115-B2-rep1
E5
WM-115 Vemurafenib Daminozide 1.0000 0.1067
uM
48
hr
1 1545 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 137.77 NGFR rabbit IgG(H+L) / donkey NGFR 1194.58
WM115-B2-rep1
E6
WM-115 Vemurafenib I-BET 1.0000 0.1067
uM
48
hr
1 1370 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 141.54 NGFR rabbit IgG(H+L) / donkey NGFR 851.57
WM115-B2-rep1
E7
WM-115 Vemurafenib Epigallocatechin gallate 1.0000 0.1067
uM
48
hr
1 1508 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 142.32 NGFR rabbit IgG(H+L) / donkey NGFR 1161.16
WM115-B2-rep1
E8
WM-115 Vemurafenib Decitabine 1.0000 0.1067
uM
48
hr
1 1358 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 155.00 NGFR rabbit IgG(H+L) / donkey NGFR 1090.08
WM115-B2-rep1
F2
WM-115 Vemurafenib Garcinol 1.0000 0.1067
uM
48
hr
1 1268 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 145.31 NGFR rabbit IgG(H+L) / donkey NGFR 1155.37
WM115-B2-rep1
F3
WM-115 Vemurafenib Pracinostat 1.0000 0.1067
uM
48
hr
1 1425 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 122.48 NGFR rabbit IgG(H+L) / donkey NGFR 911.70
WM115-B2-rep1
F4
WM-115 Vemurafenib BIX-01294 1.0000 0.1067
uM
48
hr
1 1301 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 156.60 NGFR rabbit IgG(H+L) / donkey NGFR 1057.22
WM115-B2-rep1
F5
WM-115 Vemurafenib Methylstat 1.0000 0.1067
uM
48
hr
1 1231 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 123.55 NGFR rabbit IgG(H+L) / donkey NGFR 1100.39
WM115-B2-rep1
F6
WM-115 Vemurafenib I-BET151 1.0000 0.1067
uM
48
hr
1 1232 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 134.18 NGFR rabbit IgG(H+L) / donkey NGFR 846.80
WM115-B2-rep1
F7
WM-115 Vemurafenib CX-5461 1.0000 0.1067
uM
48
hr
1 1311 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 123.99 NGFR rabbit IgG(H+L) / donkey NGFR 1203.80
WM115-B2-rep1
F8
WM-115 Vemurafenib RG-108 1.0000 0.1067
uM
48
hr
1 1171 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 137.60 NGFR rabbit IgG(H+L) / donkey NGFR 983.96
WM115-B2-rep1
G2
WM-115 Vemurafenib Anacardic acid 1.0000 0.1067
uM
48
hr
1 1092 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 137.00 NGFR rabbit IgG(H+L) / donkey NGFR 967.15
WM115-B2-rep1
G3
WM-115 Vemurafenib MC1568 1.0000 0.1067
uM
48
hr
1 1072 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 145.00 NGFR rabbit IgG(H+L) / donkey NGFR 1018.03
WM115-B2-rep1
G4
WM-115 Vemurafenib UNC0638 1.0000 0.1067
uM
48
hr
1 1111 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 130.67 NGFR rabbit IgG(H+L) / donkey NGFR 1220.72
WM115-B2-rep1
G5