5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | 1 | uM | |
| 5z-7-oxozeaenol | BCWM.1 | SYK | ISDFGLSKALR | Activation Loop | -0.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 9.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 16.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | -2.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -0.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | -10.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | 24.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 23.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | 7.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | 14.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 16.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 40.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 7.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KC1A | DIKPDNFLMGIGR | Lys2 | 32.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | -5.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 6.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | 11.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | 5.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | M4K3 | NVNTGELAAIKVIK | Lys1 | -11.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MP2K7 | DVKPSNILLDER | Lys2 | 28.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | M3K2 | ELAVKQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -9.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | -16.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MSK1_domain1 | DIKLENILLDSNGHVVLTDFGLSK | Lys2 | -5.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MK14 | QELNKTIWEVPER | Other | -8.1 | 1 | uM |