5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
5z-7-oxozeaenol BCWM.1 PIK3CD
VNWLAHNVSKDNRQ
ATP
5.1
1
uM
5z-7-oxozeaenol BCWM.1 PIK3CG
KKPLWLEFK
ATP
12.5
1
uM
5z-7-oxozeaenol BCWM.1 PIP4K2A
AKELPTLKDNDFINEGQK
ATP
14.2
1
uM
5z-7-oxozeaenol BCWM.1 FYV1
GGKSGAAFYATEDDRFILK
ATP
19.1
1
uM
5z-7-oxozeaenol BCWM.1 PITSLRE
DLKTSNLLLSHAGILK
Lys2
2.3
1
uM
5z-7-oxozeaenol BCWM.1 PKD2
DVAVKVIDK
Lys1
11.8
1
uM
5z-7-oxozeaenol BCWM.1 PKD3
DVAIKVIDK
Lys1
1
uM
5z-7-oxozeaenol BCWM.1 PKN1
VLLSEFRPSGELFAIKALK
Lys1
-24.7
1
uM
5z-7-oxozeaenol BCWM.1 PKR
DLKPSNIFLVDTK
Lys2
7.4
1
uM
5z-7-oxozeaenol BCWM.1 PLK1
CFEISDADTKEVFAGKIVPK
Lys1
1.2
1
uM
5z-7-oxozeaenol BCWM.1 PRP4
CNILHADIKPDNILVNESK
Lys2
1.7
1
uM
5z-7-oxozeaenol BCWM.1 PRPK
FLSGLELVKQGAEAR
ATP Loop
14.4
1
uM
5z-7-oxozeaenol BCWM.1 RIPK2
VQVAVKHLHIHTPLLDSER
Lys1
11.1
1
uM
5z-7-oxozeaenol BCWM.1 RIPK3
DLKPSNVLLDPELHVK
Lys2
-4.0
1
uM
5z-7-oxozeaenol BCWM.1 ROCK1,ROCK2
DVKPDNMLLDK
Lys2
22.9
1
uM
5z-7-oxozeaenol BCWM.1 RSK1 domain1
DLKPENILLDEEGHIKLTDFGLSKEAIDHEK
Lys2
12.7
1
uM
5z-7-oxozeaenol BCWM.1 RSK2 domain1
DLKPENILLDEEGHIKLTDFGLSKESIDHEK
Lys2
23.5
1
uM
5z-7-oxozeaenol BCWM.1 RSK4 domain1
DLKPENILLDEIGHIK
Lys2
25.6
1
uM
5z-7-oxozeaenol BCWM.1 SGK3
FYAVKVLQK
Lys1
-7.9
1
uM
5z-7-oxozeaenol BCWM.1 SLK
DLKAGNILFTLDGDIK
Lys2
-2.3
1
uM
5z-7-oxozeaenol BCWM.1 SMG1
DTVTIHSVGGTITILPTKTKPK
ATP
15.7
1
uM
5z-7-oxozeaenol BCWM.1 SNRK
DLKPENVVFFEK
Lys2
-11.3
1
uM
5z-7-oxozeaenol BCWM.1 SRPK1
IIHTDIKPENILLSVNEQYIR
Lys2
-1.0
1
uM
5z-7-oxozeaenol BCWM.1 STK33
DLKLENIMVK
Lys2
3.1
1
uM
5z-7-oxozeaenol BCWM.1 STLK5
YSVKVLPWLSPEVLQQNLQGYDAK
Activation Loop
-31.2
1
uM