5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
5z-7-oxozeaenol | BCWM.1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | 5.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PIK3CG | KKPLWLEFK | ATP | 12.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | 14.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | 19.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PITSLRE | DLKTSNLLLSHAGILK | Lys2 | 2.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PKD2 | DVAVKVIDK | Lys1 | 11.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PKD3 | DVAIKVIDK | Lys1 | 1 | uM | |
5z-7-oxozeaenol | BCWM.1 | PKN1 | VLLSEFRPSGELFAIKALK | Lys1 | -24.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PKR | DLKPSNIFLVDTK | Lys2 | 7.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 1.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | 1.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | PRPK | FLSGLELVKQGAEAR | ATP Loop | 14.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RIPK2 | VQVAVKHLHIHTPLLDSER | Lys1 | 11.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -4.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | ROCK1,ROCK2 | DVKPDNMLLDK | Lys2 | 22.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RSK1 domain1 | DLKPENILLDEEGHIKLTDFGLSKEAIDHEK | Lys2 | 12.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | 23.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | RSK4 domain1 | DLKPENILLDEIGHIK | Lys2 | 25.6 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SGK3 | FYAVKVLQK | Lys1 | -7.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SLK | DLKAGNILFTLDGDIK | Lys2 | -2.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | 15.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SNRK | DLKPENVVFFEK | Lys2 | -11.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | -1.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | STK33 | DLKLENIMVK | Lys2 | 3.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | -31.2 | 1 | uM |