LINCS Pilot Phase Joint Project: Sensitivity measures of six breast cancer cell lines to a library of small molecule kinase inhibitors (single drug treatments). Dataset 11 of 15: Mean cell count and mean normalized growth rate inhibition values across biological replicate 1. - Dataset (ID:20248)
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Cell | Small Molecule | Small Mol Concentration | Small Mol Conc Unit | LJP Library Plate | Timepoint | Timepoint Unit | Mean Total Cell Count Before Treatment | Mean Total Cell Count After Treatment | Mean Total Control Cell Count | Mean Relative Cell Count | Mean Normalized Growth Rate Inhibition Value |
---|---|---|---|---|---|---|---|---|---|---|---|
MCF 10A | OSI-027 | 3.33 | uM | LJP6 | 72 | hr | 513 | 1101 | 10473 | 0.1052 | 0.1917 |
MCF 10A | Pictilisib | 3.33 | uM | LJP6 | 72 | hr | 513 | 1104 | 10473 | 0.1055 | 0.1915 |
MCF7 | Canertinib | 10 | uM | LJP6 | 72 | hr | 1235 | 430 | 4056 | 0.1061 | -0.4595 |
MCF 10A | Torin1 | 1.11 | uM | LJP6 | 72 | hr | 513 | 1111 | 10473 | 0.1061 | 0.1900 |
MCF 10A | Torin1 | 0.37 | uM | LJP6 | 72 | hr | 513 | 1114 | 10473 | 0.1064 | 0.1945 |
MCF 10A | Canertinib | 0.12 | uM | LJP6 | 72 | hr | 513 | 1120 | 10473 | 0.1069 | 0.1955 |
MCF 10A | Y39983 | 10 | uM | LJP6 | 72 | hr | 513 | 1133 | 10473 | 0.1082 | 0.1992 |
MCF 10A | Selumetinib | 3.33 | uM | LJP6 | 72 | hr | 513 | 1150 | 10473 | 0.1099 | 0.2029 |
MCF 10A | NVP-AEW541 | 10 | uM | LJP5 | 72 | hr | 513 | 1146 | 10362 | 0.1106 | 0.2022 |
MCF 10A | Foretinib | 3.33 | uM | LJP5 | 72 | hr | 513 | 1147 | 10362 | 0.1107 | 0.2038 |
MCF 10A | WH-4-025 | 3.33 | uM | LJP5 | 72 | hr | 513 | 1148 | 10362 | 0.1109 | 0.2020 |
MCF 10A | Dactolisib | 10 | uM | LJP5 | 72 | hr | 513 | 1157 | 10362 | 0.1117 | 0.2062 |
MCF 10A | PD184352 | 3.33 | uM | LJP5 | 72 | hr | 513 | 1165 | 10362 | 0.1124 | 0.2079 |
MDA-MB-231 | Celastrol | 10 | uM | LJP6 | 72 | hr | 868 | 402 | 3556 | 0.1136 | -0.3153 |
MCF 10A | PF431396 | 0.37 | uM | LJP5 | 72 | hr | 513 | 1183 | 10362 | 0.1143 | 0.2122 |
MCF 10A | Alvocidib | 0.04 | uM | LJP6 | 72 | hr | 513 | 1211 | 10473 | 0.1157 | 0.2180 |
MCF 10A | AZD8055 | 0.12 | uM | LJP6 | 72 | hr | 513 | 1215 | 10473 | 0.1160 | 0.2178 |
MCF 10A | Selumetinib | 1.11 | uM | LJP6 | 72 | hr | 513 | 1235 | 10473 | 0.1180 | 0.2216 |
MCF 10A | PHA-793887 | 0.04 | uM | LJP6 | 72 | hr | 513 | 1245 | 10473 | 0.1188 | 0.2233 |
BT-20 | A443654 | 10 | uM | LJP6 | 72 | hr | 1657 | 652 | 5383 | 0.1212 | -0.4241 |
MCF 10A | Seliciclib | 10 | uM | LJP5 | 72 | hr | 513 | 1269 | 10362 | 0.1223 | 0.2294 |
MCF 10A | Barasertib | 1.11 | uM | LJP5 | 72 | hr | 513 | 1268 | 10362 | 0.1224 | 0.2319 |
MCF 10A | ZSTK474 | 10 | uM | LJP6 | 72 | hr | 513 | 1292 | 10473 | 0.1234 | 0.2346 |
MCF7 | Geldanamycin | 10 | uM | LJP5 | 72 | hr | 1235 | 525 | 4267 | 0.1234 | -0.3802 |
MCF 10A | Tozasertib | 0.12 | uM | LJP5 | 72 | hr | 513 | 1287 | 10362 | 0.1243 | 0.2362 |