Phosphorylation state and protein levels measured in BRAF(V600E/D) melanoma cell lines monitored by Reverse Phase Protein Arrays (RPPA) - Dataset (ID:20218)
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Small Molecule | Cell Line | Drug Concentration | Conc Unit | Time Point | Time Point Unit | Replicate | Scanner/Software | pMEK(S217/221) | Normalized Median pMEK(S217/221) | pERK(T202/Y204) | Normalized Median pERK(T202/Y204) | p-p90RSK(S380) | Normalized Median p-p90RSK(S380) | p-p90RSK(T573) | Normalized Median p-p90RSK(T573) | p-AKT(T308) | Normalized Median p-AKT(T308) | p-AKT(S473) | Normalized Median p-AKT(S473) | p-mTOR(S2448) | Normalized Median p-mTOR(S2448) | p-p70S6K(T421/S424) | Normalized Median p-p70S6K(T421/S424) | p-p70S6K(T389) | Normalized Median p-p70S6K(T389) | p-S6(S235/236) | Normalized Median p-S6(S235/236) | p-AMPK(T172) | Normalized Median p-AMPK(T172) | p-JNK(T183/Y185) | Normalized Median p-JNK(T183/Y185) | Total c-Jun | Normalized Median Total c-Jun | p-cJun(S63) | Normalized Median p-cJun(S63) | p-P38(T180/Y182) | Normalized Median p-P38(T180/Y182) | p-HSP27(S82) | Normalized Median p-HSP27(S82) | p-NFKB(S536) | Normalized Median p-NFKB(S536) | Bim | Normalized Median Bim | cPARP | Normalized Median cPARP | p-Histone H3(S10) | Normalized Median p-Histone H3(S10) | p27 Kip1 | Normalized Median p27 Kip1 |
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COLO 858 | 0.0000 | uM | 1 | hr | 2 | Odyssey/Microvigene | 0.5747 | 1.3514 | 0.1098 | 0.1520 | 0.1456 | 0.2342 | 0.1506 | 0.2283 | 1.0204 | 0.3906 | 0.3145 | 0.1447 | 0.1767 | 0.2033 | 0.3247 | 0.0331 | 0.0735 | 0.4367 | 0.3839 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 2 | Odyssey/Microvigene | 0.5682 | 1.1820 | 0.1148 | 0.1531 | 0.1449 | 0.2833 | 0.1621 | 0.2427 | 0.9346 | 0.3521 | 0.3040 | 0.1642 | 0.1916 | 0.2141 | 0.3521 | 0.0840 | 0.1221 | 0.4951 | 0.3712 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 2 | Odyssey/Microvigene | 0.9346 | 2.5316 | 0.1188 | 0.2132 | 0.1034 | 0.3802 | 0.1341 | 0.2717 | 1.6393 | 0.6289 | 0.4566 | 0.1610 | 0.2257 | 0.2016 | 0.3068 | 0.0565 | 0.1316 | 0.3774 | 0.5917 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 2 | Odyssey/Microvigene | 0.9524 | 2.6178 | 0.1323 | 0.1667 | 0.1280 | 0.4065 | 0.1520 | 0.2778 | 1.7422 | 0.6623 | 0.4292 | 0.1477 | 0.2212 | 0.2208 | 0.3215 | 0.1000 | 0.1287 | 0.4546 | 0.6170 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 2 | Odyssey/Microvigene | 0.6024 | 1.4006 | 0.1280 | 0.1898 | 0.1493 | 0.2519 | 0.2237 | 0.2288 | 1.0373 | 0.3774 | 0.3155 | 0.1650 | 0.1842 | 0.1773 | 0.3367 | 0.0285 | 0.0714 | 0.4049 | 0.3894 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 2 | Odyssey/Microvigene | 0.5495 | 1.2706 | 0.1357 | 0.2016 | 0.1350 | 0.2770 | 0.2268 | 0.2375 | 0.9174 | 0.3704 | 0.2817 | 0.1832 | 0.2105 | 0.1832 | 0.3718 | 0.0680 | 0.1000 | 0.4329 | 0.3687 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.8403 | 2.0833 | 0.1189 | 0.2114 | 0.1083 | 0.3333 | 0.1493 | 0.2331 | 1.6892 | 0.4902 | 0.3984 | 0.1701 | 0.2114 | 0.2033 | 0.3247 | 0.0617 | 0.1047 | 0.4098 | 0.5218 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.9615 | 2.5445 | 0.1033 | 0.2058 | 0.1224 | 0.4065 | 0.1873 | 0.2667 | 1.6051 | 0.5988 | 0.4202 | 0.1707 | 0.2203 | 0.2370 | 0.3571 | 0.0629 | 0.1342 | 0.4854 | 0.6569 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.7143 | 1.8248 | 0.1083 | 0.1567 | 0.1014 | 0.3268 | 0.1553 | 0.1992 | 1.3263 | 0.4484 | 0.3279 | 0.1412 | 0.1730 | 0.1855 | 0.2959 | 0.0400 | 0.1033 | 0.3953 | 0.4775 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.5988 | 0.9901 | 0.1161 | 0.1563 | 0.1214 | 0.2315 | 0.1543 | 0.2188 | 0.7407 | 0.3175 | 0.3345 | 0.1553 | 0.1901 | 0.2058 | 0.3195 | 0.0709 | 0.0714 | 0.4546 | 0.3539 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.8547 | 2.0080 | 0.1101 | 0.1848 | 0.0840 | 0.3690 | 0.1767 | 0.2481 | 1.5175 | 0.5291 | 0.3861 | 0.1423 | 0.2132 | 0.1597 | 0.3077 | 0.0478 | 0.1170 | 0.3356 | 0.5544 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.8772 | 2.6738 | 0.0962 | 0.1815 | 0.1071 | 0.4292 | 0.1695 | 0.2597 | 1.8083 | 0.6098 | 0.3861 | 0.1416 | 0.2119 | 0.1953 | 0.3236 | 0.0633 | 0.1166 | 0.4049 | 0.5770 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.6803 | 1.9048 | 0.1148 | 0.1504 | 0.1456 | 0.3165 | 0.1799 | 0.2439 | 1.3245 | 0.5025 | 0.3861 | 0.1543 | 0.1799 | 0.1621 | 0.3663 | 0.0166 | 0.1119 | 0.3650 | 0.4636 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 3 | Odyssey/Microvigene | 0.5556 | 1.0787 | 0.1337 | 0.1698 | 0.1454 | 0.2273 | 0.1961 | 0.2841 | 0.7634 | 0.3185 | 0.3731 | 0.1890 | 0.2262 | 0.1748 | 0.3788 | 0.0333 | 0.0787 | 0.4016 | 0.3846 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.8000 | 2.2222 | 0.1580 | 0.2375 | 0.1287 | 0.3876 | 0.1709 | 0.2793 | 1.5244 | 0.6173 | 0.5102 | 0.1812 | 0.2688 | 0.2404 | 0.3367 | 0.1155 | 0.1460 | 0.4132 | 0.5616 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.7752 | 1.9724 | 0.1536 | 0.2105 | 0.1300 | 0.4348 | 0.1724 | 0.2959 | 1.4184 | 0.6536 | 0.4854 | 0.1776 | 0.2653 | 0.2538 | 0.3597 | 0.1003 | 0.1143 | 0.5025 | 0.5495 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.6410 | 1.5221 | 0.1637 | 0.2551 | 0.1637 | 0.3257 | 0.1916 | 0.2667 | 1.3038 | 0.4878 | 0.4546 | 0.1934 | 0.2469 | 0.2299 | 0.4149 | 0.0465 | 0.0935 | 0.4975 | 0.4146 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.5917 | 1.2579 | 0.1524 | 0.2222 | 0.1718 | 0.2577 | 0.1996 | 0.2907 | 0.8475 | 0.3597 | 0.4184 | 0.2079 | 0.2564 | 0.2151 | 0.4292 | 0.0391 | 0.0800 | 0.5465 | 0.3934 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.7937 | 2.2523 | 0.1316 | 0.2092 | 0.1410 | 0.4065 | 0.1449 | 0.2801 | 1.4493 | 0.6250 | 0.4762 | 0.1761 | 0.2695 | 0.1927 | 0.3891 | 0.0518 | 0.1385 | 0.3677 | 0.5905 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.7874 | 1.9724 | 0.1570 | 0.1972 | 0.1218 | 0.4292 | 0.1686 | 0.2941 | 1.3908 | 0.6329 | 0.4464 | 0.1873 | 0.2695 | 0.1869 | 0.3953 | 0.0405 | 0.1146 | 0.4310 | 0.5725 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.6667 | 1.6779 | 0.1276 | 0.1536 | 0.1266 | 0.3086 | 0.1570 | 0.2273 | 1.5974 | 0.4854 | 0.3185 | 0.1681 | 0.1894 | 0.1621 | 0.3236 | 0.0394 | 0.0943 | 0.3831 | 0.4638 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 4 | Odyssey/Microvigene | 0.5618 | 1.2771 | 0.1229 | 0.1383 | 0.1321 | 0.2353 | 0.1639 | 0.2451 | 0.9259 | 0.3650 | 0.3077 | 0.1859 | 0.2128 | 0.1560 | 0.3322 | 0.0971 | 0.0787 | 0.4292 | 0.3689 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 5 | Odyssey/Microvigene | 0.9709 | 2.5000 | 0.1522 | 0.2151 | 0.1403 | 0.4016 | 0.1832 | 0.2786 | 1.6694 | 0.6250 | 0.5848 | 0.1876 | 0.2525 | 0.2381 | 0.3953 | 0.1351 | 0.1600 | 0.4484 | 0.6191 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 5 | Odyssey/Microvigene | 0.9804 | 2.8736 | 0.1405 | 0.2004 | 0.1513 | 0.4717 | 0.1724 | 0.3096 | 1.6026 | 0.7194 | 0.5155 | 0.1912 | 0.2762 | 0.2725 | 0.3876 | 0.1227 | 0.1233 | 0.5882 | 0.6389 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 1 | hr | 5 | Odyssey/Microvigene | 0.6452 | 1.3793 | 0.1155 | 0.1362 | 0.1258 | 0.2874 | 0.1493 | 0.1887 | 0.9804 | 0.3937 | 0.3185 | 0.1647 | 0.1838 | 0.1887 | 0.3049 | 0.0467 | 0.0787 | 0.3759 | 0.4077 |