Phosphorylation state and protein levels measured in BRAF(V600E/D) melanoma cell lines monitored by Reverse Phase Protein Arrays (RPPA) - Dataset (ID:20218)
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Small Molecule | Cell Line | Drug Concentration | Conc Unit | Time Point | Time Point Unit | Replicate | Scanner/Software | pMEK(S217/221) | Normalized Median pMEK(S217/221) | pERK(T202/Y204) | Normalized Median pERK(T202/Y204) | p-p90RSK(S380) | Normalized Median p-p90RSK(S380) | p-p90RSK(T573) | Normalized Median p-p90RSK(T573) | p-AKT(T308) | Normalized Median p-AKT(T308) | p-AKT(S473) | Normalized Median p-AKT(S473) | p-mTOR(S2448) | Normalized Median p-mTOR(S2448) | p-p70S6K(T421/S424) | Normalized Median p-p70S6K(T421/S424) | p-p70S6K(T389) | Normalized Median p-p70S6K(T389) | p-S6(S235/236) | Normalized Median p-S6(S235/236) | p-AMPK(T172) | Normalized Median p-AMPK(T172) | p-JNK(T183/Y185) | Normalized Median p-JNK(T183/Y185) | Total c-Jun | Normalized Median Total c-Jun | p-cJun(S63) | Normalized Median p-cJun(S63) | p-P38(T180/Y182) | Normalized Median p-P38(T180/Y182) | p-HSP27(S82) | Normalized Median p-HSP27(S82) | p-NFKB(S536) | Normalized Median p-NFKB(S536) | Bim | Normalized Median Bim | cPARP | Normalized Median cPARP | p-Histone H3(S10) | Normalized Median p-Histone H3(S10) | p27 Kip1 | Normalized Median p27 Kip1 |
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COLO 858 | 0.0000 | uM | 10 | hr | 8 | Odyssey/Microvigene | 0.5917 | 1.1013 | 0.1449 | 0.2268 | 0.1565 | 0.2188 | 0.2033 | 0.2416 | 0.7874 | 0.5650 | 0.3497 | 0.1567 | 0.1770 | 0.3546 | 0.3718 | 0.0787 | 0.0855 | 0.6494 | 0.4503 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 10 | hr | 8 | Odyssey/Microvigene | 0.6211 | 1.0526 | 0.1704 | 0.3175 | 0.2024 | 0.2278 | 0.2114 | 0.2475 | 0.8197 | 0.4926 | 0.5102 | 0.1748 | 0.2584 | 0.4065 | 0.4000 | 0.0746 | 0.0935 | 0.6803 | 0.4299 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 10 | hr | 8 | Odyssey/Microvigene | 0.6098 | 1.1099 | 0.1605 | 0.3448 | 0.1908 | 0.2146 | 0.2198 | 0.2695 | 0.8547 | 0.5076 | 0.4975 | 0.1686 | 0.2160 | 0.4049 | 0.4292 | 0.0488 | 0.0943 | 0.7353 | 0.4128 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 10 | hr | 8 | Odyssey/Microvigene | 0.6494 | 1.2438 | 0.1437 | 0.2028 | 0.1701 | 0.2273 | 0.1597 | 0.2165 | 0.8772 | 0.5291 | 0.3226 | 0.1482 | 0.1828 | 0.2611 | 0.3759 | 0.0847 | 0.0870 | 0.5319 | 0.4406 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 10 | hr | 8 | Odyssey/Microvigene | 0.6623 | 1.1325 | 0.1332 | 0.2075 | 0.1529 | 0.2294 | 0.1828 | 0.2364 | 0.8197 | 0.5495 | 0.3521 | 0.1582 | 0.1901 | 0.2899 | 0.4132 | 0.0794 | 0.0763 | 0.5714 | 0.4505 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 10 | hr | 8 | Odyssey/Microvigene | 0.6849 | 1.0846 | 0.1701 | 0.2577 | 0.1908 | 0.2262 | 0.1938 | 0.2591 | 0.4878 | 0.3891 | 0.1754 | 0.1938 | 0.3300 | 0.3802 | 0.0741 | 0.6536 | 0.4508 | ||||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 10 | hr | 8 | Odyssey/Microvigene | 0.6579 | 1.1312 | 0.1560 | 0.2532 | 0.1832 | 0.2037 | 0.1992 | 0.2703 | 0.9434 | 0.4902 | 0.4082 | 0.1859 | 0.2268 | 0.3279 | 0.4274 | 0.0952 | 0.7143 | 0.4293 | |||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.7874 | 1.2330 | 0.1560 | 0.2208 | 0.1698 | 0.1961 | 0.1773 | 0.2141 | 0.7246 | 0.6667 | 0.3774 | 0.1639 | 0.1698 | 0.2410 | 0.4348 | 0.1217 | 0.1156 | 0.6897 | 0.5039 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.8265 | 1.4599 | 0.1595 | 0.2092 | 0.1684 | 0.2045 | 0.1748 | 0.2222 | 0.7092 | 0.7407 | 0.3891 | 0.1553 | 0.1789 | 0.2653 | 0.4484 | 0.1258 | 0.1091 | 0.6757 | 0.5090 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.7092 | 1.0965 | 0.1957 | 0.2359 | 0.2227 | 0.1667 | 0.2058 | 0.2551 | 0.6410 | 0.5988 | 0.4762 | 0.1808 | 0.1852 | 0.3333 | 0.5780 | 0.1111 | 0.1033 | 0.7407 | 0.4632 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.8621 | 1.1403 | 0.2882 | 0.2786 | 0.1672 | 0.2469 | 0.7407 | 0.5714 | 0.5102 | 0.1996 | 0.2165 | 0.3497 | 0.5814 | 0.1449 | 0.1199 | 0.8265 | 0.5116 | ||||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.7937 | 1.2330 | 0.1473 | 0.2020 | 0.1558 | 0.1862 | 0.1815 | 0.1996 | 0.7519 | 0.6711 | 0.3731 | 0.1508 | 0.1799 | 0.2212 | 0.4016 | 0.1109 | 0.1050 | 0.6329 | 0.4700 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.8475 | 1.4577 | 0.1587 | 0.2193 | 0.1661 | 0.1927 | 0.1776 | 0.2232 | 0.7463 | 0.7246 | 0.3831 | 0.1555 | 0.1812 | 0.2463 | 0.4132 | 0.1235 | 0.1250 | 0.6536 | 0.5333 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.7042 | 1.2165 | 0.1686 | 0.2740 | 0.2037 | 0.1742 | 0.2066 | 0.2421 | 0.6494 | 0.5952 | 0.4098 | 0.1786 | 0.1949 | 0.3068 | 0.4695 | 0.1121 | 0.1214 | 0.8065 | 0.4790 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 1 | Odyssey/Microvigene | 0.8621 | 1.1173 | 0.1658 | 0.2778 | 0.2174 | 0.1767 | 0.1992 | 0.2475 | 0.7752 | 0.5650 | 0.3731 | 0.2083 | 0.2092 | 0.2899 | 0.4717 | 0.1488 | 0.1449 | 0.8065 | 0.5300 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 1.1494 | 1.9493 | 0.1681 | 0.2398 | 0.1661 | 0.2273 | 0.2123 | 0.2041 | 0.9434 | 0.9346 | 0.4717 | 0.1692 | 0.1887 | 0.2793 | 0.4167 | 0.1143 | 0.1267 | 0.6944 | 0.6191 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 1.0183 | 1.7422 | 0.1724 | 0.2398 | 0.1736 | 0.2410 | 0.1992 | 0.2237 | 0.8547 | 0.8000 | 0.4902 | 0.1689 | 0.1972 | 0.4425 | 0.1075 | 0.1174 | 0.8265 | 0.5701 | |||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 0.8772 | 1.4859 | 0.1518 | 0.1969 | 0.1761 | 0.2169 | 0.1805 | 0.2092 | 0.9259 | 0.7299 | 0.3677 | 0.1543 | 0.1565 | 0.2801 | 0.4149 | 0.0787 | 0.1370 | 0.7092 | 0.5091 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 0.7752 | 1.0834 | 0.1575 | 0.2123 | 0.1758 | 0.1783 | 0.2062 | 0.2273 | 0.7752 | 0.5556 | 0.3546 | 0.1642 | 0.1883 | 0.2755 | 0.4444 | 0.1109 | 0.1053 | 0.7463 | 0.4160 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 1.0650 | 1.8975 | 0.1595 | 0.2237 | 0.1587 | 0.2092 | 0.1832 | 0.1876 | 1.0718 | 0.8929 | 0.4065 | 0.1572 | 0.1795 | 0.4065 | 0.0901 | 0.1179 | 0.6849 | 0.6056 | |||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 0.9804 | 1.6892 | 0.1672 | 0.2183 | 0.1570 | 0.2342 | 0.1828 | 0.2070 | 1.0395 | 0.7752 | 0.3937 | 0.1541 | 0.1822 | 0.2778 | 0.4274 | 0.1339 | 0.1229 | 0.7634 | 0.6035 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 0.9259 | 1.4903 | 0.1550 | 0.2342 | 0.1996 | 0.1976 | 0.1996 | 0.2203 | 0.9434 | 0.7353 | 0.3759 | 0.1675 | 0.1707 | 0.2849 | 0.4739 | 0.0709 | 0.1221 | 0.7874 | 0.5312 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 2 | Odyssey/Microvigene | 0.7937 | 1.1455 | 0.1686 | 0.2278 | 0.1838 | 0.1848 | 0.2075 | 0.2463 | 0.7692 | 0.5405 | 0.3774 | 0.1770 | 0.1942 | 0.2688 | 0.4854 | 0.1425 | 0.0952 | 0.8000 | 0.4627 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 3 | Odyssey/Microvigene | 1.1001 | 1.8762 | 0.1629 | 0.2387 | 0.1531 | 0.2203 | 0.1942 | 0.2058 | 1.1338 | 0.8333 | 0.4444 | 0.1464 | 0.1779 | 0.2618 | 0.4167 | 0.0870 | 0.1230 | 0.6944 | 0.6314 | ||||||||||||||||||||||||
COLO 858 | 0.0000 | uM | 24 | hr | 3 | Odyssey/Microvigene | 0.9901 | 1.8519 | 0.1504 | 0.2545 | 0.1421 | 0.2193 | 0.1976 | 0.2155 | 1.0152 | 0.8065 | 0.4444 | 0.1527 | 0.1862 | 0.4630 | 0.1000 | 0.1221 | 0.8065 | 0.6558 |