Ibrutinib KiNativ -- single dose experiment - Dataset (ID:20214)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| Ibrutinib | BCWM.1 | NEK9 | DIKTLNIFLTK | Lys2 | 8.326033968 | 1 | uM |
| Ibrutinib | BCWM.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -1.255029683 | 1 | uM |
| Ibrutinib | BCWM.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 11.12523953 | 1 | uM |
| Ibrutinib | BCWM.1 | MK14 | QELNKTIWEVPER | Other | 6.71455834 | 1 | uM |
| Ibrutinib | BCWM.1 | MK11 | QELNKTVWEVPQR | Other | -0.386101983 | 1 | uM |
| Ibrutinib | BCWM.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | 0.981795646 | 1 | uM |
| Ibrutinib | BCWM.1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -80.07141375 | 1 | uM |
| Ibrutinib | BCWM.1 | KS6B2 | DLKPENIMLSSQGHIK | Lys2 | -25.23123498 | 1 | uM |
| Ibrutinib | BCWM.1 | PAN3 | VMDPTKILITGK | ATP | -19.88546356 | 1 | uM |
| Ibrutinib | BCWM.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | -14.73329296 | 1 | uM |
| Ibrutinib | BCWM.1 | PDK1 | EYAIKILEK | Lys1 | -26.37271999 | 1 | uM |
| Ibrutinib | BCWM.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | -23.81656725 | 1 | uM |
| Ibrutinib | BCWM.1 | CDK14 | LVALKVIR | Lys1 | -8.300309889 | 1 | uM |
| Ibrutinib | BCWM.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | -23.59607344 | 1 | uM |
| Ibrutinib | BCWM.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | -19.55661054 | 1 | uM |
| Ibrutinib | BCWM.1 | PI4KB | VPHTQAVVLNSKDK | ATP | -2.264791249 | 1 | uM |
| Ibrutinib | BCWM.1 | PIK3C2B | VIFKCGDDLRQDMLTLQMIR | ATP | -5.03638468 | 1 | uM |
| Ibrutinib | BCWM.1 | PIK3C3 | TEDGGKYPVIFKHGDDLR | ATP | -4.759272068 | 1 | uM |
| Ibrutinib | BCWM.1 | PIK3CB | VFGEDSVGVIFKNGDDLRQDMLTLQMLR | ATP | -25.58117019 | 1 | uM |
| Ibrutinib | BCWM.1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | -5.232559785 | 1 | uM |
| Ibrutinib | BCWM.1 | PIK3CG | KKPLWLEFK | ATP | 24.89529253 | 1 | uM |
| Ibrutinib | BCWM.1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | -5.492209336 | 1 | uM |
| Ibrutinib | BCWM.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | -37.02302597 | 1 | uM |
| Ibrutinib | BCWM.1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | -3.050757538 | 1 | uM |
| Ibrutinib | BCWM.1 | PITSLRE | DLKTSNLLLSHAGILK | Lys2 | 0.867558432 | 1 | uM |