JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JNK-IN-8 | A-375 | DNAPK | kGGSWIQEINVAEK | ATP | 12.8 | 1 | uM |
| JNK-IN-8 | A-375 | eEF2K | YIkYNSNSGFVRDDNIR | Protein Kinase Domain | 10.0 | 1 | uM |
| JNK-IN-8 | A-375 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -5.4 | 1 | uM |
| JNK-IN-8 | A-375 | EGFR | IPVAIkELR | Lys1 | 0.1 | 1 | uM |
| JNK-IN-8 | A-375 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 1.4 | 1 | uM |
| JNK-IN-8 | A-375 | MK03 | YIHSANVLHRDLkPSNLLINTTCDLK | Lys2 | 28.3 | 1 | uM |
| JNK-IN-8 | A-375 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 0.2 | 1 | uM |
| JNK-IN-8 | A-375 | Erk5 | DLkPSNLLVNENCELK | Lys2 | -4.7 | 1 | uM |
| JNK-IN-8 | A-375 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | -16.6 | 1 | uM |
| JNK-IN-8 | A-375 | FER | QEDGGVYSSSGLkQIPIKWTAPEALNYGR | Activation Loop | -1.4 | 1 | uM |
| JNK-IN-8 | A-375 | FER | DKTSVAVkTCKEDLPQELK | Lys1 | 13.9 | 1 | uM |
| JNK-IN-8 | A-375 | FER | TSVAVkTCKEDLPQELK | Lys1 | -7.0 | 1 | uM |
| JNK-IN-8 | A-375 | FRAP1 | IQSIAPSLQVITSkQRPR | -6.5 | 1 | uM | |
| JNK-IN-8 | A-375 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 7.9 | 1 | uM |
| JNK-IN-8 | A-375 | GCK | DTVTSELAAVkIVK | Lys1 | -20.4 | 1 | uM |
| JNK-IN-8 | A-375 | GCK | DIkGANLLLTLQGDVK | Lys2 | 10.4 | 1 | uM |
| JNK-IN-8 | A-375 | GCN2_domain2 | VQNKLDGCCYAVkR | Lys1 | 9.0 | 1 | uM |
| JNK-IN-8 | A-375 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | -32.8 | 1 | uM |
| JNK-IN-8 | A-375 | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | 10.6 | 1 | uM |
| JNK-IN-8 | A-375 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | -8.5 | 1 | uM |
| JNK-IN-8 | A-375 | IKKA | IIHRDLkPENIVLQDVGGK | Lys2 | -3.4 | 1 | uM |
| JNK-IN-8 | A-375 | IKKA | DLkPENIVLQDVGGK | Lys2 | 4.9 | 1 | uM |
| JNK-IN-8 | A-375 | IKKB | IIHRDLkPENIVLQQGEQR | Lys2 | 36.2 | 1 | uM |
| JNK-IN-8 | A-375 | IKKB | DLkPENIVLQQGEQR | Lys2 | -6.5 | 1 | uM |
| JNK-IN-8 | A-375 | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | 12.2 | 1 | uM |