OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
OTSSP167 MDA-MB-468 RSK2_domain2
DLKPSNILYVDESGNPESIR
Lys2
>97
1
uM
OTSSP167 MDA-MB-468 RSKL1_domain1
VLGVIDKVLLVMDTR
ATP
-41.3
1
uM
OTSSP167 MDA-MB-468 SGK3
FYAVKVLQK
Lys1
91.5
1
uM
OTSSP167 MDA-MB-468 SLK
DLKAGNILFTLDGDIK
Lys2
93.4
1
uM
OTSSP167 MDA-MB-468 SMG1
DTVTIHSVGGTITILPTKTKPK
ATP
98.1
1
uM
OTSSP167 MDA-MB-468 SNRK
DLKPENVVFFEK
Lys2
12.8
1
uM
OTSSP167 MDA-MB-468 SRPK1
IIHTDIKPENILLSVNEQYIR
Lys2
86.8
1
uM
OTSSP167 MDA-MB-468 SRPK1/2
FVAMKVVK
Lys1
72.8
1
uM
OTSSP167 MDA-MB-468 STLK5
YSVKVLPWLSPEVLQQNLQGYDAK
Activation Loop
83.5
1
uM
OTSSP167 MDA-MB-468 SYK
ISDFGLSKALR
Activation Loop
91.6
1
uM
OTSSP167 MDA-MB-468 MAP3K7,TAK1
DLKPPNLLLVAGGTVLK
Lys2
>93
1
uM
OTSSP167 MDA-MB-468 TAO1,TAOK3
DIKAGNILLTEPGQVK
Lys2
>99
1
uM
OTSSP167 MDA-MB-468 TAOK2
DVKAGNILLSEPGLVK
Lys2
>97
1
uM
OTSSP167 MDA-MB-468 TBK1
TGDLFAIKVFNNISFLRPVDVQMR
Lys1
>90
1
uM
OTSSP167 MDA-MB-468 TLK1
YLNEIKPPIIHYDLKPGNILLVDGTACGEIK
Lys2
53.7
1
uM
OTSSP167 MDA-MB-468 TLK1/2
YLNEIKPPIIHYDLKPGNILLVNGTACGEIK
Lys2
16.7
1
uM
OTSSP167 MDA-MB-468 TNK1
SVPVAVKSLR
Lys1
>95
1
uM
OTSSP167 MDA-MB-468 ULK1
DLKPQNILLSNPAGR
Lys2
-64.2
1
uM
OTSSP167 MDA-MB-468 ULK3
NISHLDLKPQNILLSSLEKPHLK
Lys2
75.3
1
uM
OTSSP167 MDA-MB-468 Wnk1,Wnk2,Wnk3
DLKCDNIFITGPTGSVK
Lys2
12.6
1
uM
OTSSP167 MDA-MB-468 MLTK
WISQDKEVAVKK
Lys1
>98
1
uM
OTSSP167 MDA-MB-468 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIKGQNVLLTENAEVK
Lys2
>98
1
uM
OTSSP167 MDA-MB-468 KCC2D
IPTGQEYAAKIINTKK
Lys1
93.1
1
uM
OTSSP167 MDA-MB-468 CDK20
DLKPANLLISASGQLK
Lys2
81.5
1
uM
OTSSP167 MDA-MB-468 KC1G2
DVKPENFLVGRPGTK
Lys2
89.7
1
uM