QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 STLK5
YSVKVLPWLSPEVLQQNLQGYDAK
Activation Loop
29.01675643
1
uM
QL-XII-47 BCWM.1 STLK6
HTPTGTLVTIKITNLENCNEER
Lys1
ND
1
uM
QL-XII-47 BCWM.1 SYK
ISDFGLSKALR
Activation Loop
7.40661852
1
uM
QL-XII-47 BCWM.1 MAP3K7,TAK1
DLKPPNLLLVAGGTVLK
Lys2
-8.438191166
1
uM
QL-XII-47 BCWM.1 TAO1,TAOK3
DIKAGNILLTEPGQVK
Lys2
-11.78552859
1
uM
QL-XII-47 BCWM.1 TAOK2
DVKAGNILLSEPGLVK
Lys2
-25.18845999
1
uM
QL-XII-47 BCWM.1 TBK1
TGDLFAIKVFNNISFLRPVDVQMR
Lys1
16.75925379
1
uM
QL-XII-47 BCWM.1 TEC
YVLDDQYTSSSGAKFPVK
Activation Loop
70.24556535
1
uM
QL-XII-47 BCWM.1 TLK1
YLNEIKPPIIHYDLKPGNILLVDGTACGEIK
Lys2
11.52268187
1
uM
QL-XII-47 BCWM.1 TLK1/2
YLNEIKPPIIHYDLKPGNILLVNGTACGEIK
Lys2
-3.9573695
1
uM
QL-XII-47 BCWM.1 ULK1
DLKPQNILLSNPAGR
Lys2
10.00533539
1
uM
QL-XII-47 BCWM.1 ULK3
NISHLDLKPQNILLSSLEKPHLK
Lys2
10.43573458
1
uM
QL-XII-47 BCWM.1 VRK2
MLDVLEYIHENEYVHGDIKAANLLLGYK
Lys2
-1.787209636
1
uM
QL-XII-47 BCWM.1 WEE1
YIHSMSLVHMDIKPSNIFISR
Lys2
0.899795474
1
uM
QL-XII-47 BCWM.1 Wnk1,Wnk2,Wnk3
DLKCDNIFITGPTGSVK
Lys2
-6.796460792
1
uM
QL-XII-47 BCWM.1 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIKGQNVLLTENAEVK
Lys2
-19.55134985
1
uM
QL-XII-47 BCWM.1 ZC2/TNIK
TGQLAAIKVMDVTGDEEEEIKQEINMLKK
Lys1
4.081055995
1
uM
QL-XII-47 BCWM.1 BLK
IIDSEYTAQEGAKFPIK
Activation Loop
47.0732956
1
uM
QL-XII-47 BCWM.1 KCC2D
IPTGQEYAAKIINTKK
Lys1
0.853020424
1
uM
QL-XII-47 BCWM.1 KCC4
DLKPENLLYATPAPDAPLK
Lys2
-28.81450984
1
uM
QL-XII-47 BCWM.1 KC1G2
DVKPENFLVGRPGTK
Lys2
-6.736083059
1
uM
QL-XII-47 BCWM.1 EPHB1
YLQDDTSDPTYTSSLGGKIPVR
Activation Loop
-4.242361482
1
uM
QL-XII-47 BCWM.1 MK01
DLKPSNLLLNTTCDLK
Lys2
0.422779704
1
uM
QL-XII-47 BCWM.1 FRK
HEIKLPVK
Activation Loop
-7.289586984
1
uM
QL-XII-47 BCWM.1 KSR1
SKNVFYDNGKVVITDFGLFGISGVVR
Activation Loop
-16.59423638
1
uM