QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 29.01675643 | 1 | uM |
QL-XII-47 | BCWM.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | ND | 1 | uM |
QL-XII-47 | BCWM.1 | SYK | ISDFGLSKALR | Activation Loop | 7.40661852 | 1 | uM |
QL-XII-47 | BCWM.1 | MAP3K7,TAK1 | DLKPPNLLLVAGGTVLK | Lys2 | -8.438191166 | 1 | uM |
QL-XII-47 | BCWM.1 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | -11.78552859 | 1 | uM |
QL-XII-47 | BCWM.1 | TAOK2 | DVKAGNILLSEPGLVK | Lys2 | -25.18845999 | 1 | uM |
QL-XII-47 | BCWM.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 16.75925379 | 1 | uM |
QL-XII-47 | BCWM.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 70.24556535 | 1 | uM |
QL-XII-47 | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 11.52268187 | 1 | uM |
QL-XII-47 | BCWM.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -3.9573695 | 1 | uM |
QL-XII-47 | BCWM.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | 10.00533539 | 1 | uM |
QL-XII-47 | BCWM.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 10.43573458 | 1 | uM |
QL-XII-47 | BCWM.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | -1.787209636 | 1 | uM |
QL-XII-47 | BCWM.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 0.899795474 | 1 | uM |
QL-XII-47 | BCWM.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -6.796460792 | 1 | uM |
QL-XII-47 | BCWM.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | -19.55134985 | 1 | uM |
QL-XII-47 | BCWM.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 4.081055995 | 1 | uM |
QL-XII-47 | BCWM.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | 47.0732956 | 1 | uM |
QL-XII-47 | BCWM.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 0.853020424 | 1 | uM |
QL-XII-47 | BCWM.1 | KCC4 | DLKPENLLYATPAPDAPLK | Lys2 | -28.81450984 | 1 | uM |
QL-XII-47 | BCWM.1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | -6.736083059 | 1 | uM |
QL-XII-47 | BCWM.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | -4.242361482 | 1 | uM |
QL-XII-47 | BCWM.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 0.422779704 | 1 | uM |
QL-XII-47 | BCWM.1 | FRK | HEIKLPVK | Activation Loop | -7.289586984 | 1 | uM |
QL-XII-47 | BCWM.1 | KSR1 | SKNVFYDNGKVVITDFGLFGISGVVR | Activation Loop | -16.59423638 | 1 | uM |