QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | MWCL.1 | MAP3K3 | ELASKQVQFDPDSPETSKEVSALECEIQLLK | Lys1 | -1.791203787 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | 16.84992087 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | -9.625870933 | 1 | uM |
QL-XII-47 | MWCL.1 | MARK2,MARK3 | DLKAENLLLDADMNIK | Lys2 | -11.86915829 | 1 | uM |
QL-XII-47 | MWCL.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 10.94267365 | 1 | uM |
QL-XII-47 | MWCL.1 | MARK3,MARK4 | EVAIKIIDK | Lys1 | 5.793943076 | 1 | uM |
QL-XII-47 | MWCL.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | -89.96758232 | 1 | uM |
QL-XII-47 | MWCL.1 | MAST3 | DLKPDNLLITSLGHIK | Lys2 | 3.312930204 | 1 | uM |
QL-XII-47 | MWCL.1 | MASTL | GAFGKVYLGQK | ATP Loop | -5.128672656 | 1 | uM |
QL-XII-47 | MWCL.1 | MASTL | LYAVKVVK | Lys1 | -4.9183009 | 1 | uM |
QL-XII-47 | MWCL.1 | MLK3 | DLKSNNILLLQPIESDDMEHK | Lys2 | 24.61377493 | 1 | uM |
QL-XII-47 | MWCL.1 | MLK4 | DLKSSNILLLEK | Lys2 | ND | 1 | uM |
QL-XII-47 | MWCL.1 | MLKL | APVAIKVFK | Lys1 | 7.351746937 | 1 | uM |
QL-XII-47 | MWCL.1 | MSK1_domain1 | DIKLENILLDSNGHVVLTDFGLSK | Lys2 | -16.80838137 | 1 | uM |
QL-XII-47 | MWCL.1 | MSK2 domain1 | DLKLENVLLDSEGHIVLTDFGLSK | Lys2 | -60.55728513 | 1 | uM |
QL-XII-47 | MWCL.1 | MST1 | ETGQIVAIKQVPVESDLQEIIK | Lys1 | 15.40673657 | 1 | uM |
QL-XII-47 | MWCL.1 | MST2 | ESGQVVAIKQVPVESDLQEIIK | Lys1 | 16.41617398 | 1 | uM |
QL-XII-47 | MWCL.1 | MST3 | DIKAANVLLSEHGEVK | Lys2 | 3.17261014 | 1 | uM |
QL-XII-47 | MWCL.1 | MST4 | TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK | Lys1 | -3.541851435 | 1 | uM |
QL-XII-47 | MWCL.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | -0.541351906 | 1 | uM |
QL-XII-47 | MWCL.1 | MYO3A,MYO3B | DVKGNNILLTTEGGVK | Lys2 | 5.489365936 | 1 | uM |
QL-XII-47 | MWCL.1 | NDR1 | DIKPDNLLLDSK | Lys2 | 0.686324454 | 1 | uM |
QL-XII-47 | MWCL.1 | NDR2 | DIKPDNLLLDAK | Lys2 | 13.19299985 | 1 | uM |
QL-XII-47 | MWCL.1 | NEK1 | DIKSQNIFLTK | Lys2 | 0.042103767 | 1 | uM |
QL-XII-47 | MWCL.1 | NEK3 | SKNIFLTQNGK | Activation Loop | 9.919741065 | 1 | uM |