QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 MWCL.1 MAP3K3
ELASKQVQFDPDSPETSKEVSALECEIQLLK
Lys1
-1.791203787
1
uM
QL-XII-47 MWCL.1 MAP3K4
DIKGANIFLTSSGLIK
Lys2
16.84992087
1
uM
QL-XII-47 MWCL.1 MAP3K5
DIKGDNVLINTYSGVLK
Lys2
-9.625870933
1
uM
QL-XII-47 MWCL.1 MARK2,MARK3
DLKAENLLLDADMNIK
Lys2
-11.86915829
1
uM
QL-XII-47 MWCL.1 MARK3
EVAIKIIDKTQLNPTSLQK
Lys1
10.94267365
1
uM
QL-XII-47 MWCL.1 MARK3,MARK4
EVAIKIIDK
Lys1
5.793943076
1
uM
QL-XII-47 MWCL.1 MAST1,MAST2
DLKPDNLLITSMGHIK
Lys2
-89.96758232
1
uM
QL-XII-47 MWCL.1 MAST3
DLKPDNLLITSLGHIK
Lys2
3.312930204
1
uM
QL-XII-47 MWCL.1 MASTL
GAFGKVYLGQK
ATP Loop
-5.128672656
1
uM
QL-XII-47 MWCL.1 MASTL
LYAVKVVK
Lys1
-4.9183009
1
uM
QL-XII-47 MWCL.1 MLK3
DLKSNNILLLQPIESDDMEHK
Lys2
24.61377493
1
uM
QL-XII-47 MWCL.1 MLK4
DLKSSNILLLEK
Lys2
ND
1
uM
QL-XII-47 MWCL.1 MLKL
APVAIKVFK
Lys1
7.351746937
1
uM
QL-XII-47 MWCL.1 MSK1_domain1
DIKLENILLDSNGHVVLTDFGLSK
Lys2
-16.80838137
1
uM
QL-XII-47 MWCL.1 MSK2 domain1
DLKLENVLLDSEGHIVLTDFGLSK
Lys2
-60.55728513
1
uM
QL-XII-47 MWCL.1 MST1
ETGQIVAIKQVPVESDLQEIIK
Lys1
15.40673657
1
uM
QL-XII-47 MWCL.1 MST2
ESGQVVAIKQVPVESDLQEIIK
Lys1
16.41617398
1
uM
QL-XII-47 MWCL.1 MST3
DIKAANVLLSEHGEVK
Lys2
3.17261014
1
uM
QL-XII-47 MWCL.1 MST4
TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK
Lys1
-3.541851435
1
uM
QL-XII-47 MWCL.1 MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
-0.541351906
1
uM
QL-XII-47 MWCL.1 MYO3A,MYO3B
DVKGNNILLTTEGGVK
Lys2
5.489365936
1
uM
QL-XII-47 MWCL.1 NDR1
DIKPDNLLLDSK
Lys2
0.686324454
1
uM
QL-XII-47 MWCL.1 NDR2
DIKPDNLLLDAK
Lys2
13.19299985
1
uM
QL-XII-47 MWCL.1 NEK1
DIKSQNIFLTK
Lys2
0.042103767
1
uM
QL-XII-47 MWCL.1 NEK3
SKNIFLTQNGK
Activation Loop
9.919741065
1
uM