QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | PKD2 | DVAVKVIDK | Lys1 | -4.298882666 | 1 | uM |
QL-XII-47 | BCWM.1 | PKD3 | DVAIKVIDK | Lys1 | 28.45310221 | 1 | uM |
QL-XII-47 | BCWM.1 | PKN1 | VLLSEFRPSGELFAIKALK | Lys1 | 32.0802275 | 1 | uM |
QL-XII-47 | BCWM.1 | PKR | DLKPSNIFLVDTK | Lys2 | 1.597115102 | 1 | uM |
QL-XII-47 | BCWM.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 10.38740966 | 1 | uM |
QL-XII-47 | BCWM.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | -20.14127866 | 1 | uM |
QL-XII-47 | BCWM.1 | PRPK | FLSGLELVKQGAEAR | ATP Loop | -5.388379383 | 1 | uM |
QL-XII-47 | BCWM.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -37.08301629 | 1 | uM |
QL-XII-47 | BCWM.1 | RAF1 | DMKSNNIFLHEGLTVK | Lys2 | -4.024800041 | 1 | uM |
QL-XII-47 | BCWM.1 | RIPK2 | VQVAVKHLHIHTPLLDSER | Lys1 | -40.21606445 | 1 | uM |
QL-XII-47 | BCWM.1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | -9.173875348 | 1 | uM |
QL-XII-47 | BCWM.1 | ROCK1,ROCK2 | DVKPDNMLLDK | Lys2 | 19.88680143 | 1 | uM |
QL-XII-47 | BCWM.1 | RSK1 domain1 | DLKPENILLDEEGHIKLTDFGLSKEAIDHEK | Lys2 | -58.92112884 | 1 | uM |
QL-XII-47 | BCWM.1 | RSK1_domain2 | DLKPSNILYVDESGNPECLR | Lys2 | 3.780249297 | 1 | uM |
QL-XII-47 | BCWM.1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | -52.47434469 | 1 | uM |
QL-XII-47 | BCWM.1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | 6.304020294 | 1 | uM |
QL-XII-47 | BCWM.1 | RSK3_domain1 | DLKPENILLDEEGHIKITDFGLSK | Lys2 | -54.52802421 | 1 | uM |
QL-XII-47 | BCWM.1 | RSK4 domain1 | DLKPENILLDEIGHIK | Lys2 | -43.35732659 | 1 | uM |
QL-XII-47 | BCWM.1 | RSKL1_domain1 | VLGVIDKVLLVMDTR | ATP | 46.48841594 | 1 | uM |
QL-XII-47 | BCWM.1 | SGK3 | FYAVKVLQK | Lys1 | 7.055655022 | 1 | uM |
QL-XII-47 | BCWM.1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 30.24247402 | 1 | uM |
QL-XII-47 | BCWM.1 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | -2.926780018 | 1 | uM |
QL-XII-47 | BCWM.1 | SNRK | DLKPENVVFFEK | Lys2 | 24.94063876 | 1 | uM |
QL-XII-47 | BCWM.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | 0.388055572 | 1 | uM |
QL-XII-47 | BCWM.1 | SRPK1/2 | FVAMKVVK | Lys1 | 17.54405997 | 1 | uM |