TAE-684 KINOMEscan - Dataset (ID:20199)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| NVP-TAE684 | DCAMKL2 | 16.0 | nM |
| NVP-TAE684 | DCAMKL3 | 14.0 | nM |
| NVP-TAE684 | DDR1 | 140.0 | nM |
| NVP-TAE684 | DDR2 | 4100.0 | nM |
| NVP-TAE684 | M3K12 | 42.0 | nM |
| NVP-TAE684 | DMPK | 2100.0 | nM |
| NVP-TAE684 | DMPK2 | 9500.0 | nM |
| NVP-TAE684 | DRAK1 | 2900.0 | nM |
| NVP-TAE684 | DRAK2 | 7100.0 | nM |
| NVP-TAE684 | DYRK1A | 2900.0 | nM |
| NVP-TAE684 | DYRK1B | 4500.0 | nM |
| NVP-TAE684 | DYRK2 | nM | |
| NVP-TAE684 | EGFR | 180.0 | nM |
| NVP-TAE684 | EGFR(E746-A750del) | 81.0 | nM |
| NVP-TAE684 | EGFR(G719C) | 2000.0 | nM |
| NVP-TAE684 | EGFR(G719S) | 1600.0 | nM |
| NVP-TAE684 | EGFR(L747-E749del, A750P) | 72.0 | nM |
| NVP-TAE684 | EGFR(L747-S752del, P753S) | 110.0 | nM |
| NVP-TAE684 | EGFR(L747-T751del,Sins) | 79.0 | nM |
| NVP-TAE684 | EGFR(L858R) | 46.0 | nM |
| NVP-TAE684 | EGFR(L858R,T790M) | 3.4 | nM |
| NVP-TAE684 | EGFR(L861Q) | 98.0 | nM |
| NVP-TAE684 | EGFR(S752-I759del) | 400.0 | nM |
| NVP-TAE684 | EGFR(T790M) | 7.1 | nM |
| NVP-TAE684 | EIF2AK1 | nM |