TAE-684 KINOMEscan - Dataset (ID:20199)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| NVP-TAE684 | AAK1 | 470.0 | nM |
| NVP-TAE684 | ABL1(E255K)-phosphorylated | 190.0 | nM |
| NVP-TAE684 | ABL1(F317I)-nonphosphorylated | 93.0 | nM |
| NVP-TAE684 | ABL1(F317I)-phosphorylated | 14.0 | nM |
| NVP-TAE684 | ABL1(F317L)-nonphosphorylated | 54.0 | nM |
| NVP-TAE684 | ABL1(F317L)-phosphorylated | 19.0 | nM |
| NVP-TAE684 | ABL1(H396P)-nonphosphorylated | 73.0 | nM |
| NVP-TAE684 | ABL1(H396P)-phosphorylated | 160.0 | nM |
| NVP-TAE684 | ABL1(M351T)-phosphorylated | 95.0 | nM |
| NVP-TAE684 | ABL1(Q252H)-nonphosphorylated | 39.0 | nM |
| NVP-TAE684 | ABL1(Q252H)-phosphorylated | 70.0 | nM |
| NVP-TAE684 | ABL1(T315I)-nonphosphorylated | 52.0 | nM |
| NVP-TAE684 | ABL1(T315I)-phosphorylated | 5.4 | nM |
| NVP-TAE684 | ABL1(Y253F)-phosphorylated | 100.0 | nM |
| NVP-TAE684 | ABL1-nonphosphorylated | 200.0 | nM |
| NVP-TAE684 | ABL1-phosphorylated | 170.0 | nM |
| NVP-TAE684 | ABL2 | 380.0 | nM |
| NVP-TAE684 | ACVR1 | 29.0 | nM |
| NVP-TAE684 | ACVR1B | 97.0 | nM |
| NVP-TAE684 | ACVR2A | 2200.0 | nM |
| NVP-TAE684 | ACVR2B | 4300.0 | nM |
| NVP-TAE684 | ACVRL1 | 57.0 | nM |
| NVP-TAE684 | ADCK3 | 1700.0 | nM |
| NVP-TAE684 | ADCK4 | 92.0 | nM |
| NVP-TAE684 | AKT1 | nM |