TAE-684 KINOMEscan - Dataset (ID:20199)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
NVP-TAE684 | PRKX | 5800.0 | nM |
NVP-TAE684 | PRP4 | 7600.0 | nM |
NVP-TAE684 | FAK2 | 1.1 | nM |
NVP-TAE684 | SIK3 | 1300.0 | nM |
NVP-TAE684 | RAF1 | nM | |
NVP-TAE684 | RET | 150.0 | nM |
NVP-TAE684 | RET(M918T) | 140.0 | nM |
NVP-TAE684 | RET(V804L) | 120.0 | nM |
NVP-TAE684 | RET(V804M) | 140.0 | nM |
NVP-TAE684 | RIOK1 | nM | |
NVP-TAE684 | RIOK2 | nM | |
NVP-TAE684 | RIOK3 | 3500.0 | nM |
NVP-TAE684 | RIPK1 | nM | |
NVP-TAE684 | RIPK2 | 9600.0 | nM |
NVP-TAE684 | RIPK4 | 3200.0 | nM |
NVP-TAE684 | RIPK5 | 57.0 | nM |
NVP-TAE684 | ROCK1 | 37.0 | nM |
NVP-TAE684 | ROCK2 | 130.0 | nM |
NVP-TAE684 | ROS1 | 0.5 | nM |
NVP-TAE684 | RPS6KA4(Kin.Dom.1-N-terminal) | 2500.0 | nM |
NVP-TAE684 | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
NVP-TAE684 | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
NVP-TAE684 | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
NVP-TAE684 | RSK1(Kin.Dom.1-N-terminal) | 160.0 | nM |
NVP-TAE684 | RSK1(Kin.Dom.2-C-terminal) | 650.0 | nM |