VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Tozasertib | DCAMKL2 | nM | |
| Tozasertib | DCAMKL3 | 3600.0 | nM |
| Tozasertib | DDR1 | 28.0 | nM |
| Tozasertib | DDR2 | 230.0 | nM |
| Tozasertib | M3K12 | 190.0 | nM |
| Tozasertib | DMPK | nM | |
| Tozasertib | DMPK2 | nM | |
| Tozasertib | DRAK1 | 9000.0 | nM |
| Tozasertib | DRAK2 | nM | |
| Tozasertib | DYRK1A | nM | |
| Tozasertib | DYRK1B | nM | |
| Tozasertib | DYRK2 | nM | |
| Tozasertib | EGFR | nM | |
| Tozasertib | EGFR(E746-A750del) | nM | |
| Tozasertib | EGFR(G719C) | nM | |
| Tozasertib | EGFR(G719S) | nM | |
| Tozasertib | EGFR(L747-E749del, A750P) | nM | |
| Tozasertib | EGFR(L747-S752del, P753S) | nM | |
| Tozasertib | EGFR(L747-T751del,Sins) | nM | |
| Tozasertib | EGFR(L858R) | nM | |
| Tozasertib | EGFR(L858R,T790M) | nM | |
| Tozasertib | EGFR(L861Q) | nM | |
| Tozasertib | EGFR(S752-I759del) | nM | |
| Tozasertib | EGFR(T790M) | nM | |
| Tozasertib | EIF2AK1 | nM |