VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Tozasertib | PRKX | nM | |
| Tozasertib | PRP4 | 2500.0 | nM |
| Tozasertib | FAK2 | 2600.0 | nM |
| Tozasertib | SIK3 | nM | |
| Tozasertib | RAF1 | nM | |
| Tozasertib | RET | 28.0 | nM |
| Tozasertib | RET(M918T) | 26.0 | nM |
| Tozasertib | RET(V804L) | 8.6 | nM |
| Tozasertib | RET(V804M) | 13.0 | nM |
| Tozasertib | RIOK1 | 360.0 | nM |
| Tozasertib | RIOK2 | 250.0 | nM |
| Tozasertib | RIOK3 | 600.0 | nM |
| Tozasertib | RIPK1 | 20.0 | nM |
| Tozasertib | RIPK2 | nM | |
| Tozasertib | RIPK4 | 300.0 | nM |
| Tozasertib | RIPK5 | nM | |
| Tozasertib | ROCK1 | nM | |
| Tozasertib | ROCK2 | nM | |
| Tozasertib | ROS1 | 610.0 | nM |
| Tozasertib | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
| Tozasertib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
| Tozasertib | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
| Tozasertib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
| Tozasertib | RSK1(Kin.Dom.1-N-terminal) | 7900.0 | nM |
| Tozasertib | RSK1(Kin.Dom.2-C-terminal) | nM |