VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tozasertib | ABL1(E255K)-phosphorylated | 3.0 | nM |
Tozasertib | ABL1(H396P)-phosphorylated | 3.1 | nM |
Tozasertib | ABL1(H396P)-nonphosphorylated | 3.3 | nM |
Tozasertib | ABL1(Q252H)-nonphosphorylated | 3.8 | nM |
Tozasertib | AURKA | 3.9 | nM |
Tozasertib | ABL2 | 4.0 | nM |
Tozasertib | FLT3(N841I) | 4.3 | nM |
Tozasertib | FLT3(K663Q) | 4.8 | nM |
Tozasertib | ABL1(M351T)-phosphorylated | 5.3 | nM |
Tozasertib | AURKC | 6.3 | nM |
Tozasertib | FLT3 | 6.5 | nM |
Tozasertib | AURKB | 7.4 | nM |
Tozasertib | ABL1-phosphorylated | 7.5 | nM |
Tozasertib | ABL1(Y253F)-phosphorylated | 7.8 | nM |
Tozasertib | RET(V804L) | 8.6 | nM |
Tozasertib | PLK4 | 9.2 | nM |
Tozasertib | ABL1(T315I)-phosphorylated | 9.3 | nM |
Tozasertib | ABL1(Q252H)-phosphorylated | 9.4 | nM |
Tozasertib | ABL1(T315I)-nonphosphorylated | 9.7 | nM |
Tozasertib | ABL1-nonphosphorylated | 13.0 | nM |
Tozasertib | RET(V804M) | 13.0 | nM |
Tozasertib | FLT3(D835H) | 14.0 | nM |
Tozasertib | MLCK | 15.0 | nM |
Tozasertib | RIPK1 | 20.0 | nM |
Tozasertib | RET(M918T) | 26.0 | nM |